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TargetRas-related C3 botulinum toxin substrate 1
LigandBDBM54561
Substrate/Competitorn/a
Meas. Tech.Oxadiazole SAR compounds tested via Multiplex dose response to identify specific small molecule inhibitors of Ras and Ras-related GTPases specifically Rac1 activated mutant
Ki 180±n/a nM
Citation PubChem, PC Oxadiazole SAR compounds tested via Multiplex dose response to identify specific small molecule inhibitors of Ras and Ras-related GTPases specifically Rac1 activated mutant PubChem Bioassay(2009)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Ras-related C3 botulinum toxin substrate 1
Name:Ras-related C3 botulinum toxin substrate 1
Synonyms:RAC1_MOUSE | Rac1 | Rac1 protein
Type:PROTEIN
Mol. Mass.:21455.91
Organism:Mus musculus
Description:EBI_101485
Residue:192
Sequence:
MQAIKCVVVGDGAVGKTCLLISYTTNAFPGEYIPTVFDNYSANVMVDGKPVNLGLWDTAG
QEDYDRLRPLSYPQTDVFLICFSLVSPASFENVRAKWYPEVRHHCPNTPIILVGTKLDLR
DDKDTIEKLKEKKLTPITYPQGLAMAKEIGAVKYLECSALTQRGLKTVFDEAIRAVLCPP
PVKKRKRKCLLL
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BDBM54561
n/a
NameBDBM54561
Synonyms:3-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-1-[4-[2-(trifluoromethyl)phenyl]-1-piperazinyl]-1-propanone | 3-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-1-[4-[2-(trifluoromethyl)phenyl]piperazin-1-yl]propan-1-one | 3-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-1-[4-[2-(trifluoromethyl)phenyl]piperazino]propan-1-one | KUC103372N | UNM-0000306082 | cid_42596909
TypeSmall organic molecule
Emp. Form.C23H23F3N4O3
Mol. Mass.460.4489
SMILESCOc1ccc(cc1)-c1noc(CCC(=O)N2CCN(CC2)c2ccccc2C(F)(F)F)n1
Structure
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