| Reaction Details |
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 | Report a problem with these data |
| Target | Ras-related C3 botulinum toxin substrate 1 |
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| Ligand | BDBM54571 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Oxadiazole SAR compounds tested via Multiplex dose response to identify specific small molecule inhibitors of Ras and Ras-related GTPases specifically Rac1 activated mutant |
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| Ki | 80±n/a nM |
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| Citation |  PubChem, PC Oxadiazole SAR compounds tested via Multiplex dose response to identify specific small molecule inhibitors of Ras and Ras-related GTPases specifically Rac1 activated mutant PubChem Bioassay(2009)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| |
| Ras-related C3 botulinum toxin substrate 1 |
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| Name: | Ras-related C3 botulinum toxin substrate 1 |
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| Synonyms: | RAC1_MOUSE | Rac1 | Rac1 protein |
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| Type: | PROTEIN |
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| Mol. Mass.: | 21455.91 |
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| Organism: | Mus musculus |
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| Description: | EBI_101485 |
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| Residue: | 192 |
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| Sequence: | MQAIKCVVVGDGAVGKTCLLISYTTNAFPGEYIPTVFDNYSANVMVDGKPVNLGLWDTAG
QEDYDRLRPLSYPQTDVFLICFSLVSPASFENVRAKWYPEVRHHCPNTPIILVGTKLDLR
DDKDTIEKLKEKKLTPITYPQGLAMAKEIGAVKYLECSALTQRGLKTVFDEAIRAVLCPP
PVKKRKRKCLLL
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| BDBM54571 |
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| n/a |
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| Name | BDBM54571 |
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| Synonyms: | 1-[4-(4-fluorophenyl)-1-piperazinyl]-3-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-1-propanone | 1-[4-(4-fluorophenyl)piperazin-1-yl]-3-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]propan-1-one | 1-[4-(4-fluorophenyl)piperazino]-3-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]propan-1-one | KUC103398N | UNM-0000306115 | cid_42628041 |
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| Type | Small organic molecule |
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| Emp. Form. | C22H23FN4O3 |
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| Mol. Mass. | 410.4414 |
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| SMILES | COc1ccc(cc1)-c1noc(CCC(=O)N2CCN(CC2)c2ccc(F)cc2)n1 |
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| Structure | 
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