| Reaction Details |
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 | Report a problem with these data |
| Target | Metabotropic glutamate receptor 4 [Q124R] |
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| Ligand | BDBM55090 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Modulation of the Metabotropic Glutamate Receptor mGluR4: Rat PAM Potency |
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| EC50 | 250±n/a nM |
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| Citation |  PubChem, PC Modulation of the Metabotropic Glutamate Receptor mGluR4: Rat PAM Potency PubChem Bioassay(2010)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| Metabotropic glutamate receptor 4 [Q124R] |
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| Name: | Metabotropic glutamate receptor 4 [Q124R] |
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| Synonyms: | GRM4_RAT | Gprc1d | Grm4 | Mglur4 | glutamate receptor, metabotropic 4 precursor |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 101878.86 |
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| Organism: | Rattus norvegicus |
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| Description: | gi_12083595 |
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| Residue: | 912 |
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| Sequence: | MSGKGGWAWWWARLPLCLLLSLYAPWVPSSLGKPKGHPHMNSIRIDGDITLGGLFPVHGR
GSEGKACGELKKEKGIHRLEAMLFALDRINNDPDLLPNITLGARILDTCSRDTHALEQSL
TFVRALIEKDGTEVRCGSGGPPIITKPERVVGVIGASGSSVSIMVANILRLFKIPQISYA
STAPDLSDNSRYDFFSRVVPSDTYQAQAMVDIVRALKWNYVSTLASEGSYGESGVEAFIQ
KSRENGGVCIAQSVKIPREPKTGEFDKIIKRLLETSNARGIIIFANEDDIRRVLEAARRA
NQTGHFFWMGSDSWGSKSAPVLRLEEVAEGAVTILPKRMSVRGFDRYFSSRTLDNNRRNI
WFAEFWEDNFHCKLSRHALKKGSHIKKCTNRERIGQDSAYEQEGKVQFVIDAVYAMGHAL
HAMHRDLCPGRVGLCPRMDPVDGTQLLKYIRNVNFSGIAGNPVTFNENGDAPGRYDIYQY
QLRNGSAEYKVIGSWTDHLHLRIERMQWPGSGQQLPRSICSLPCQPGERKKTVKGMACCW
HCEPCTGYQYQVDRYTCKTCPYDMRPTENRTSCQPIPIVKLEWDSPWAVLPLFLAVVGIA
ATLFVVVTFVRYNDTPIVKASGRELSYVLLAGIFLCYATTFLMIAEPDLGTCSLRRIFLG
LGMSISYAALLTKTNRIYRIFEQGKRSVSAPRFISPASQLAITFILISLQLLGICVWFVV
DPSHSVVDFQDQRTLDPRFARGVLKCDISDLSLICLLGYSMLLMVTCTVYAIKTRGVPET
FNEAKPIGFTMYTTCIVWLAFIPIFFGTSQSADKLYIQTTTLTVSVSLSASVSLGMLYMP
KVYIILFHPEQNVPKRKRSLKAVVTAATMSNKFTQKGNFRPNGEAKSELCENLETPALAT
KQTYVTYTNHAI
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| BDBM55090 |
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| n/a |
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| Name | BDBM55090 |
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| Synonyms: | VU0404304-2 | cid_46869948 |
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| Type | Small organic molecule |
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| Emp. Form. | C22H18ClN3O3 |
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| Mol. Mass. | 407.85 |
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| SMILES | [H][C@@]12C(C(=O)N(C1=O)c1ccc(NC(=O)c3ccccn3)cc1Cl)[C@@]1([H])CC[C@]2([H])C=C1 |c:34,TLB:6:1:27.26:30.31,THB:3:2:27.26:30.31| |
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| Structure | 
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