| Reaction Details |
|---|
 | Report a problem with these data |
| Target | M18 aspartyl aminopeptidase |
|---|
| Ligand | BDBM34340 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | QFRET-based biochemical high throughput dose response assay for inhibitors of the Plasmodium falciparum M18 Aspartyl Aminopeptidase (PFM18AAP). |
|---|
| IC50 | 4284±n/a nM |
|---|
| Citation |  PubChem, PC QFRET-based biochemical high throughput dose response assay for inhibitors of the Plasmodium falciparum M18 Aspartyl Aminopeptidase (PFM18AAP). PubChem Bioassay(2009)[AID] |
|---|
| More Info.: | Get all data from this article, Solution Info, Assay Method |
|---|
| |
| M18 aspartyl aminopeptidase |
|---|
| Name: | M18 aspartyl aminopeptidase |
|---|
| Synonyms: | n/a |
|---|
| Type: | Enzyme Catalytic Domain |
|---|
| Mol. Mass.: | 65642.43 |
|---|
| Organism: | Plasmodium falciparum 3D7 |
|---|
| Description: | gi_23505220 |
|---|
| Residue: | 570 |
|---|
| Sequence: | MDKKAREYAQDALKFIQRSGSNFLACKNLKERLENNGFINLSEGETWNLNKNEGYVLCKE
NRNICGFFVGKNFNIDTGSILISIGHIDSCALKISPNNNVIKKKIHQINVECYGSGLWHT
WFDRSLGLSGQVLYKKGNKLVEKLIQINKSVLFLPSLAIHLQNRTRYDFSVKINYENHIK
PIISTTLFNQLNKCKRNNVHHDTILTTDTKFSHKENSQNKRDDQMCHSFNDKDVSNHNLD
KNTIEHLTNQQNEEKNKHTKDNPNSKDIVEHINTDNSYPLLYLLSKELNCKEEDILDFEL
CLMDTQEPCFTGVYEEFIEGARFDNLLGSFCVFEGFIELVNSIKNHTSNENTNHTNNITN
DINDNIHNNLYISIGYDHEEIGSLSEVGARSYCTKNFIDRIISSVFKKEIHEKNLSVQEI
YGNLVNRSFILNVDMAHCSHPNYPETVQDNHQLFFHEGIAIKYNTNKNYVTSPLHASLIK
RTFELYYNKYKQQIKYQNFMVKNDTPCGSTVGSMVAANLSMPGIDIGIPQLAMHSIREIA
AVHDVFFLIKGVFAFYTYYNQVLSTCVHDK
|
|
|
|---|
| BDBM34340 |
|---|
| n/a |
|---|
| Name | BDBM34340 |
|---|
| Synonyms: | 2-(4-methyl-3-piperidin-1-ylsulfonyl-phenyl)-1,2-benzothiazol-3-one | 2-(4-methyl-3-piperidin-1-ylsulfonylphenyl)-1,2-benzothiazol-3-one | 2-(4-methyl-3-piperidinosulfonyl-phenyl)-1,2-benzothiazol-3-one | 2-[4-methyl-3-(1-piperidinylsulfonyl)phenyl]-1,2-benzothiazol-3-one | MLS000057572 | SMR000060796 | cid_2327953 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C19H20N2O3S2 |
|---|
| Mol. Mass. | 388.504 |
|---|
| SMILES | Cc1ccc(cc1S(=O)(=O)N1CCCCC1)-n1sc2ccccc2c1=O |
|---|
| Structure | 
|
|---|
Search and Browse
