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TargetKallikrein-5
LigandBDBM32697
Substrate/Competitorn/a
Meas. Tech.Kallikrein 5 1536 HTS Dose Response Confirmation
IC50 852.39±n/a nM
Citation PubChem, PC Kallikrein 5 1536 HTS Dose Response Confirmation PubChem Bioassay(2008)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Kallikrein-5
Name:Kallikrein-5
Synonyms:KLK5 | KLK5_HUMAN | Kallikrein 5 | SCTE | kallikrein-related peptidase 5 preproprotein
Type:PROTEIN
Mol. Mass.:32031.72
Organism:Homo sapiens (Human)
Description:EBI_12584
Residue:293
Sequence:
MATARPPWMWVLCALITALLLGVTEHVLANNDVSCDHPSNTVPSGSNQDLGAGAGEDARS
DDSSSRIINGSDCDMHTQPWQAALLLRPNQLYCGAVLVHPQWLLTAAHCRKKVFRVRLGH
YSLSPVYESGQQMFQGVKSIPHPGYSHPGHSNDLMLIKLNRRIRPTKDVRPINVSSHCPS
AGTKCLVSGWGTTKSPQVHFPKVLQCLNISVLSQKRCEDAYPRQIDDTMFCAGDKAGRDS
CQGDSGGPVVCNGSLQGLVSWGDYPCARPNRPGVYTNLCKFTKWIQETIQANS
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BDBM32697
n/a
NameBDBM32697
Synonyms:(3-Furan-2-yl-5-methylsulfanyl-[1,2,4]triazol-1-yl)-phenyl-methanone | MLS000527913 | SMR000120487 | [3-(2-furanyl)-5-(methylthio)-1,2,4-triazol-1-yl]-phenylmethanone | [3-(2-furyl)-5-(methylthio)-1,2,4-triazol-1-yl]-phenyl-methanone | [3-(furan-2-yl)-5-methylsulfanyl-1,2,4-triazol-1-yl]-phenyl-methanone | [3-(furan-2-yl)-5-methylsulfanyl-1,2,4-triazol-1-yl]-phenylmethanone | cid_1088427
TypeSmall organic molecule
Emp. Form.C14H11N3O2S
Mol. Mass.285.321
SMILESCSc1nc(nn1C(=O)c1ccccc1)-c1ccco1
Structure
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