Reaction Details |
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Target | Calmodulin-1 |
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Ligand | BDBM59169 |
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Substrate/Competitor | n/a |
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Meas. Tech. | Fluorescence spectroscopy |
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Kd | 1.0e+4±n/a nM |
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Citation | Trevitt, CR; Craven, CJ; Milanesi, L; Syson, K; Mattinen, ML; Perkins, J; Annila, A; Hunter, CA; Waltho, JP Enhanced ligand affinity for receptors in which components of the binding site are independently mobile. Chem Biol12:89-97 (2005) [PubMed] Article |
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More Info.: | Get all data from this article, Assay Method |
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Calmodulin-1 |
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Name: | Calmodulin-1 |
Synonyms: | CALM | CALM1 | CALM1_HUMAN | CALM2 | CAM | CAM1 | CAM2 | CAMB | Calmodulin-2 |
Type: | Protein |
Mol. Mass.: | 16813.73 |
Organism: | Human |
Description: | P0DP23 |
Residue: | 149 |
Sequence: | MADQLTEEQIAEFKEAFSLFDKDGDGTITTKELGTVMRSLGQNPTEAELQDMINEVDADG
NGTIDFPEFLTMMARKMKDTDSEEEIREAFRVFDKDGNGYISAAELRHVMTNLGEKLTDE
EVDEMIREADIDGDGQVNYEEFVQMMTAK
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BDBM59169 |
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n/a |
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Name | BDBM59169 |
Synonyms: | BT1 |
Type | Small organic molecule |
Emp. Form. | C34H32N2O6 |
Mol. Mass. | 564.6277 |
SMILES | COC(=O)[C@@H](CC(=O)c1cccc(c1)C(=O)C[C@@H](Cc1c[nH]c2ccccc12)C(=O)OC)Cc1c[nH]c2ccccc12 |r| |
Structure |
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