| Reaction Details |
|---|
 | Report a problem with these data |
| Target | M17 leucyl aminopeptidase |
|---|
| Ligand | BDBM59994 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | Inhibitors of Plasmodium falciparum M17- Family Leucine Aminopeptidase (M17LAP) |
|---|
| IC50 | 1020±n/a nM |
|---|
| Citation |  PubChem, PC Inhibitors of Plasmodium falciparum M17- Family Leucine Aminopeptidase (M17LAP) PubChem Bioassay(2009)[AID] |
|---|
| More Info.: | Get all data from this article, Solution Info, Assay Method |
|---|
| |
| M17 leucyl aminopeptidase |
|---|
| Name: | M17 leucyl aminopeptidase |
|---|
| Synonyms: | leucine aminopeptidase |
|---|
| Type: | Enzyme Catalytic Domain |
|---|
| Mol. Mass.: | 67834.32 |
|---|
| Organism: | Plasmodium falciparum 3D7 |
|---|
| Description: | gi_124809582 |
|---|
| Residue: | 605 |
|---|
| Sequence: | MYFSSLCKFLPISEKEKIYLNIVKKRFCKSNIYYNNNNNNIINYNKRGLKFYPFCNNLKK
NINFVNINNKKGINFHSINKERKMASEVPQVVSLDPTSIPIEYNTPIHDIKVQVYDIKGG
CNVEEGLTIFLVNNPGKENGPVKISSKVNDKNVSEFLKDENMEKFNVKLGTSKHFYMFND
NKNSVAVGYVGCGSVADLSEADMKRVVLSLVTMLHDNKLSKLTVVFEINVDKNLFRFFLE
TLFYEYMTDERFKSTDKNVNMEYIKHLGVYINNADTYKEEVEKARVYYFGTYYASQLIAA
PSNYCNPVSLSNAAVELAQKLNLEYKILGVKELEELKMGAYLSVGKGSMYPNKFIHLTYK
SKGDVKKKIALVGKGITFDSGGYNLKAAPGSMIDLMKFDMSGCAAVLGCAYCVGTLKPEN
VEIHFLSAVCENMVSKNSYRPGDIITASNGKTIEVGNTDAEGRLTLADALVYAEKLGVDY
IVDIATLTGAMLYSLGTSYAGVFGNNEELINKILNSSKTSNEPVWWLPIINEYRATLNSK
YADINNISSSVKASSIVASLFLKEFVQNTAWAHIDIAGVSWNFKARKPKGFGVRLLTEFV
LNDAL
|
|
|
|---|
| BDBM59994 |
|---|
| n/a |
|---|
| Name | BDBM59994 |
|---|
| Synonyms: | 6-[[4-(4-chloranylphenoxy)phenyl]carbamoyl]cyclohex-3-ene-1-carboxylic acid | 6-[[4-(4-chlorophenoxy)anilino]-oxomethyl]-1-cyclohex-3-enecarboxylic acid | 6-[[4-(4-chlorophenoxy)phenyl]carbamoyl]cyclohex-3-ene-1-carboxylic acid | 6-{[4-(4-chlorophenoxy)anilino]carbonyl}-3-cyclohexene-1-carboxylic acid | MLS000704600 | SMR000231117 | cid_4990949 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C20H18ClNO4 |
|---|
| Mol. Mass. | 371.814 |
|---|
| SMILES | OC(=O)C1CC=CCC1C(=O)Nc1ccc(Oc2ccc(Cl)cc2)cc1 |c:5| |
|---|
| Structure | 
|
|---|
Search and Browse
