| Reaction Details |
|---|
 | Report a problem with these data |
| Target | M17 leucyl aminopeptidase |
|---|
| Ligand | BDBM60016 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | Inhibitors of Plasmodium falciparum M17- Family Leucine Aminopeptidase (M17LAP) |
|---|
| IC50 | 1000±n/a nM |
|---|
| Citation |  PubChem, PC Inhibitors of Plasmodium falciparum M17- Family Leucine Aminopeptidase (M17LAP) PubChem Bioassay(2009)[AID] |
|---|
| More Info.: | Get all data from this article, Solution Info, Assay Method |
|---|
| |
| M17 leucyl aminopeptidase |
|---|
| Name: | M17 leucyl aminopeptidase |
|---|
| Synonyms: | leucine aminopeptidase |
|---|
| Type: | Enzyme Catalytic Domain |
|---|
| Mol. Mass.: | 67834.32 |
|---|
| Organism: | Plasmodium falciparum 3D7 |
|---|
| Description: | gi_124809582 |
|---|
| Residue: | 605 |
|---|
| Sequence: | MYFSSLCKFLPISEKEKIYLNIVKKRFCKSNIYYNNNNNNIINYNKRGLKFYPFCNNLKK
NINFVNINNKKGINFHSINKERKMASEVPQVVSLDPTSIPIEYNTPIHDIKVQVYDIKGG
CNVEEGLTIFLVNNPGKENGPVKISSKVNDKNVSEFLKDENMEKFNVKLGTSKHFYMFND
NKNSVAVGYVGCGSVADLSEADMKRVVLSLVTMLHDNKLSKLTVVFEINVDKNLFRFFLE
TLFYEYMTDERFKSTDKNVNMEYIKHLGVYINNADTYKEEVEKARVYYFGTYYASQLIAA
PSNYCNPVSLSNAAVELAQKLNLEYKILGVKELEELKMGAYLSVGKGSMYPNKFIHLTYK
SKGDVKKKIALVGKGITFDSGGYNLKAAPGSMIDLMKFDMSGCAAVLGCAYCVGTLKPEN
VEIHFLSAVCENMVSKNSYRPGDIITASNGKTIEVGNTDAEGRLTLADALVYAEKLGVDY
IVDIATLTGAMLYSLGTSYAGVFGNNEELINKILNSSKTSNEPVWWLPIINEYRATLNSK
YADINNISSSVKASSIVASLFLKEFVQNTAWAHIDIAGVSWNFKARKPKGFGVRLLTEFV
LNDAL
|
|
|
|---|
| BDBM60016 |
|---|
| n/a |
|---|
| Name | BDBM60016 |
|---|
| Synonyms: | 2-[(4-keto-1H-benzofuro[3,2-d]pyrimidin-2-yl)thio]-N-(3-methoxyphenyl)acetamide | MLS000697289 | N-(3-methoxyphenyl)-2-[(4-oxidanylidene-1H-[1]benzofuro[3,2-d]pyrimidin-2-yl)sulfanyl]ethanamide | N-(3-methoxyphenyl)-2-[(4-oxo-1H-[1]benzofuro[3,2-d]pyrimidin-2-yl)sulfanyl]acetamide | N-(3-methoxyphenyl)-2-[(4-oxo-1H-benzofuro[3,2-d]pyrimidin-2-yl)thio]acetamide | SMR000237965 | cid_2141294 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C19H15N3O4S |
|---|
| Mol. Mass. | 381.405 |
|---|
| SMILES | COc1cccc(NC(=O)CSc2nc3c4ccccc4oc3c(=O)[nH]2)c1 |
|---|
| Structure | 
|
|---|
Search and Browse
