| Reaction Details |
|---|
 | Report a problem with these data |
| Target | M17 leucyl aminopeptidase |
|---|
| Ligand | BDBM60055 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | Inhibitors of Plasmodium falciparum M17- Family Leucine Aminopeptidase (M17LAP) |
|---|
| IC50 | 1200±n/a nM |
|---|
| Citation |  PubChem, PC Inhibitors of Plasmodium falciparum M17- Family Leucine Aminopeptidase (M17LAP) PubChem Bioassay(2009)[AID] |
|---|
| More Info.: | Get all data from this article, Solution Info, Assay Method |
|---|
| |
| M17 leucyl aminopeptidase |
|---|
| Name: | M17 leucyl aminopeptidase |
|---|
| Synonyms: | leucine aminopeptidase |
|---|
| Type: | Enzyme Catalytic Domain |
|---|
| Mol. Mass.: | 67834.32 |
|---|
| Organism: | Plasmodium falciparum 3D7 |
|---|
| Description: | gi_124809582 |
|---|
| Residue: | 605 |
|---|
| Sequence: | MYFSSLCKFLPISEKEKIYLNIVKKRFCKSNIYYNNNNNNIINYNKRGLKFYPFCNNLKK
NINFVNINNKKGINFHSINKERKMASEVPQVVSLDPTSIPIEYNTPIHDIKVQVYDIKGG
CNVEEGLTIFLVNNPGKENGPVKISSKVNDKNVSEFLKDENMEKFNVKLGTSKHFYMFND
NKNSVAVGYVGCGSVADLSEADMKRVVLSLVTMLHDNKLSKLTVVFEINVDKNLFRFFLE
TLFYEYMTDERFKSTDKNVNMEYIKHLGVYINNADTYKEEVEKARVYYFGTYYASQLIAA
PSNYCNPVSLSNAAVELAQKLNLEYKILGVKELEELKMGAYLSVGKGSMYPNKFIHLTYK
SKGDVKKKIALVGKGITFDSGGYNLKAAPGSMIDLMKFDMSGCAAVLGCAYCVGTLKPEN
VEIHFLSAVCENMVSKNSYRPGDIITASNGKTIEVGNTDAEGRLTLADALVYAEKLGVDY
IVDIATLTGAMLYSLGTSYAGVFGNNEELINKILNSSKTSNEPVWWLPIINEYRATLNSK
YADINNISSSVKASSIVASLFLKEFVQNTAWAHIDIAGVSWNFKARKPKGFGVRLLTEFV
LNDAL
|
|
|
|---|
| BDBM60055 |
|---|
| n/a |
|---|
| Name | BDBM60055 |
|---|
| Synonyms: | 6-({[3-(methoxycarbonyl)-4-(4-methylphenyl)-2-thienyl]amino}carbonyl)-3-cyclohexene-1-carboxylic acid | 6-[[3-carbomethoxy-4-(p-tolyl)-2-thienyl]carbamoyl]cyclohex-3-ene-1-carboxylic acid | 6-[[3-methoxycarbonyl-4-(4-methylphenyl)thiophen-2-yl]carbamoyl]cyclohex-3-ene-1-carboxylic acid | 6-[[[3-methoxycarbonyl-4-(4-methylphenyl)-2-thiophenyl]amino]-oxomethyl]-1-cyclohex-3-enecarboxylic acid | MLS000704820 | SMR000231287 | cid_4066105 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C21H21NO5S |
|---|
| Mol. Mass. | 399.46 |
|---|
| SMILES | COC(=O)c1c(NC(=O)C2CC=CCC2C(O)=O)scc1-c1ccc(C)cc1 |c:11| |
|---|
| Structure | 
|
|---|
Search and Browse
