| Reaction Details |
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 | Report a problem with these data |
| Target | M17 leucyl aminopeptidase |
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| Ligand | BDBM53916 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Inhibitors of Plasmodium falciparum M17- Family Leucine Aminopeptidase (M17LAP) |
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| IC50 | 1000±n/a nM |
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| Citation |  PubChem, PC Inhibitors of Plasmodium falciparum M17- Family Leucine Aminopeptidase (M17LAP) PubChem Bioassay(2009)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| M17 leucyl aminopeptidase |
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| Name: | M17 leucyl aminopeptidase |
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| Synonyms: | leucine aminopeptidase |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 67834.32 |
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| Organism: | Plasmodium falciparum 3D7 |
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| Description: | gi_124809582 |
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| Residue: | 605 |
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| Sequence: | MYFSSLCKFLPISEKEKIYLNIVKKRFCKSNIYYNNNNNNIINYNKRGLKFYPFCNNLKK
NINFVNINNKKGINFHSINKERKMASEVPQVVSLDPTSIPIEYNTPIHDIKVQVYDIKGG
CNVEEGLTIFLVNNPGKENGPVKISSKVNDKNVSEFLKDENMEKFNVKLGTSKHFYMFND
NKNSVAVGYVGCGSVADLSEADMKRVVLSLVTMLHDNKLSKLTVVFEINVDKNLFRFFLE
TLFYEYMTDERFKSTDKNVNMEYIKHLGVYINNADTYKEEVEKARVYYFGTYYASQLIAA
PSNYCNPVSLSNAAVELAQKLNLEYKILGVKELEELKMGAYLSVGKGSMYPNKFIHLTYK
SKGDVKKKIALVGKGITFDSGGYNLKAAPGSMIDLMKFDMSGCAAVLGCAYCVGTLKPEN
VEIHFLSAVCENMVSKNSYRPGDIITASNGKTIEVGNTDAEGRLTLADALVYAEKLGVDY
IVDIATLTGAMLYSLGTSYAGVFGNNEELINKILNSSKTSNEPVWWLPIINEYRATLNSK
YADINNISSSVKASSIVASLFLKEFVQNTAWAHIDIAGVSWNFKARKPKGFGVRLLTEFV
LNDAL
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|
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| BDBM53916 |
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| n/a |
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| Name | BDBM53916 |
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| Synonyms: | 2-[2-[(7-ethyl-[1,3]dioxolo[4,5-g]quinolin-6-yl)sulfanyl]ethanoylamino]-4,5-dimethoxy-benzoic acid | 2-[[2-[(7-ethyl-[1,3]dioxolo[4,5-g]quinolin-6-yl)sulfanyl]acetyl]amino]-4,5-dimethoxybenzoic acid | 2-[[2-[(7-ethyl-[1,3]dioxolo[4,5-g]quinolin-6-yl)thio]-1-oxoethyl]amino]-4,5-dimethoxybenzoic acid | 2-[[2-[(7-ethyl-[1,3]dioxolo[4,5-g]quinolin-6-yl)thio]acetyl]amino]-4,5-dimethoxy-benzoic acid | MLS000714808 | SMR000274787 | cid_3208264 |
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| Type | Small organic molecule |
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| Emp. Form. | C23H22N2O7S |
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| Mol. Mass. | 470.495 |
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| SMILES | CCc1cc2cc3OCOc3cc2nc1SCC(=O)Nc1cc(OC)c(OC)cc1C(O)=O |
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| Structure | 
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