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| Reaction Details | |||
|---|---|---|---|
 | Report a problem with these data | ||
| Target | Regulator of G-protein signaling 8 | ||
| Ligand | BDBM47732 | ||
| Substrate/Competitor | n/a | ||
| Meas. Tech. | Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS8-Galphao for SAR Compounds | ||
| EC50 | 3681±n/a nM | ||
| Citation |  PubChem, PC Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS8-Galphao for SAR Compounds PubChem Bioassay(2010)[AID] | ||
| More Info.: | Get all data from this article, Solution Info, Assay Method | ||
| Regulator of G-protein signaling 8 | |||
| Name: | Regulator of G-protein signaling 8 | ||
| Synonyms: | RGS8 | RGS8_HUMAN | Regulator of G-protein signaling 8 (RGS8) | ||
| Type: | Enzyme Catalytic Domain | ||
| Mol. Mass.: | 20925.80 | ||
| Organism: | Homo sapiens (Human) | ||
| Description: | gi_74355113 | ||
| Residue: | 180 | ||
| Sequence: |
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| BDBM47732 | |||
| n/a | |||
| Name | BDBM47732 | ||
| Synonyms: | 2,6,7-trihydroxy-9-o-phenetyl-fluorone | 9-(2-ethoxyphenyl)-2,6,7-trihydroxy-3-xanthenone | 9-(2-ethoxyphenyl)-2,6,7-trihydroxy-3H-xanthen-3-one | 9-(2-ethoxyphenyl)-2,6,7-trihydroxyxanthen-3-one | 9-(2-ethoxyphenyl)-2,6,7-tris(oxidanyl)xanthen-3-one | MLS000578271 | SMR000197680 | cid_2931388 | ||
| Type | Small organic molecule | ||
| Emp. Form. | C21H16O6 | ||
| Mol. Mass. | 364.3481 | ||
| SMILES | CCOc1ccccc1-c1c2cc(O)c(O)cc2oc2cc(=O)c(O)cc12 |(13.35,3.58,;13.35,2.04,;12.01,1.27,;10.68,2.04,;10.68,3.58,;9.35,4.35,;8.01,3.58,;8.01,2.04,;9.35,1.27,;9.35,-.27,;10.68,-1.04,;12.06,-.22,;13.45,-1.01,;14.78,-.24,;13.45,-2.62,;14.78,-3.39,;12.06,-3.41,;10.68,-2.58,;9.35,-3.35,;8.01,-2.58,;6.63,-3.41,;5.24,-2.62,;3.91,-3.39,;5.24,-1.01,;3.91,-.24,;6.63,-.22,;8.01,-1.04,)| | ||
| Structure | 
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