Reaction Details |
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Target | Regulator of G-protein signaling 19 |
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Ligand | BDBM47747 |
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Substrate/Competitor | n/a |
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Meas. Tech. | Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS19-Galphao for SAR Compounds |
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EC50 | 30000±n/a nM |
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Citation | PubChem, PC Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS19-Galphao for SAR Compounds PubChem Bioassay(2010)[AID] |
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More Info.: | Get all data from this article, Solution Info, Assay Method |
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Regulator of G-protein signaling 19 |
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Name: | Regulator of G-protein signaling 19 |
Synonyms: | G protein signalling regulator 19 | GAIP | GNAI3IP | RGS19 | RGS19_HUMAN | Regulator of G-protein signaling 19 (RGS19) |
Type: | Enzyme Catalytic Domain |
Mol. Mass.: | 24631.38 |
Organism: | Homo sapiens (Human) |
Description: | gi_86990435 |
Residue: | 217 |
Sequence: | MPTPHEAEKQITGPEEADRPPSMSSHDTASPAAPSRNPCCLCWCCCCSCSWNQERRRAWQ
ASRESKLQPLPSCEVCATPSPEEVQSWAQSFDKLMHSPAGRSVFRAFLRTEYSEENMLFW
LACEELKAEANQHVVDEKARLIYEDYVSILSPKEVSLDSRVREGINKKMQEPSAHTFDDA
QLQIYTLMHRDSYPRFLSSPTYRALLLQGPSQSSSEA
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BDBM47747 |
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n/a |
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Name | BDBM47747 |
Synonyms: | 4-[(E)-[3-[3-(diethylsulfamoyl)phenyl]-5-thioxo-1H-1,2,4-triazol-4-yl]iminomethyl]benzoic acid methyl ester | 4-[[3-[3-(diethylsulfamoyl)phenyl]-5-sulfanylidene-1H-1,2,4-triazol-4-yl]iminomethyl]benzoic acid methyl ester | 4-[[3-[3-(diethylsulfamoyl)phenyl]-5-thioxo-1H-1,2,4-triazol-4-yl]iminomethyl]benzoic acid methyl ester | MLS000408811 | SMR000243078 | cid_2387418 | methyl 4-[[3-[3-(diethylsulfamoyl)phenyl]-5-sulfanylidene-1H-1,2,4-triazol-4-yl]iminomethyl]benzoate |
Type | Small organic molecule |
Emp. Form. | C21H23N5O4S2 |
Mol. Mass. | 473.568 |
SMILES | CCN(CC)S(=O)(=O)c1cccc(c1)-c1n[nH]c(=S)n1N=Cc1ccc(cc1)C(=O)OC |w:20.21| |
Structure |
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