Ki Summary

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Target

Epstein-Barr nuclear antigen 1

Ligand

BDBM62498

Substrate/Competitor

n/a

Meas. Tech.

Fluorescence polarization-based biochemical high throughput dose response assay for inhibitors of the Epstein-Barr virus nuclear antigen 1 (EBNA-1)

IC50

6913±n/a nM

Citation

PubChem, PC Fluorescence polarization-based biochemical high throughput dose response assay for inhibitors of the Epstein-Barr virus nuclear antigen 1 (EBNA-1) PubChem Bioassay(2010)[AID]

More Info.:

Get all data from this article, Solution Info, Assay Method

Epstein-Barr nuclear antigen 1

Name:

Epstein-Barr nuclear antigen 1

Synonyms:

EBNA-1 protein | EBNA1 | EBNA1_EBVB9 | Epstein-Barr virus protease (EBV Pr)

Type:

Enzyme Catalytic Domain

Mol. Mass.:

56444.81

Organism:

Human herpesvirus 4

Description:

gi_23893623

Residue:

641

Sequence:

MSDEGPGTGPGNGLGEKGDTSGPEGSGGSGPQRRGGDNHGRGRGRGRGRGGGRPGAPGGS
GSGPRHRDGVRRPQKRPSCIGCKGTHGGTGAGAGAGGAGAGGAGAGGGAGAGGGAGGAGG
AGGAGAGGGAGAGGGAGGAGGAGAGGGAGAGGGAGGAGAGGGAGGAGGAGAGGGAGAGGG
AGGAGAGGGAGGAGGAGAGGGAGAGGAGGAGGAGAGGAGAGGGAGGAGGAGAGGAGAGGA
GAGGAGAGGAGGAGAGGAGGAGAGGAGGAGAGGGAGGAGAGGGAGGAGAGGAGGAGAGGA
GGAGAGGAGGAGAGGGAGAGGAGAGGGGRGRGGSGGRGRGGSGGRGRGGSGGRRGRGRER
ARGGSRERARGRGRGRGEKRPRSPSSQSSSSGSPPRRPPPGRRPFFHPVGEADYFEYHQE
GGPDGEPDVPPGAIEQGPADDPGEGPSTGPRGQGDGGRRKKGGWFGKHRGQGGSNPKFEN
IAEGLRALLARSHVERTTDEGTWVAGVFVYGGSKTSLYNLRRGTALAIPQCRLTPLSRLP
FGMAPGPGPQPGPLRESIVCYFMVFLQTHIFAEVLKDAIKDLVMTKPAPTCNIRVTVCSF
DDGVDLPPWFPPMVEGAAAEGDDGDDGDEGGDGDEGEEGQE

BDBM62498

n/a

Name

BDBM62498

Synonyms:

2-cyclopropyl-5-[4-[4-(3-methoxyphenyl)piperazin-1-yl]sulfonylphenyl]-1,3-oxazole | 2-cyclopropyl-5-[4-[4-(3-methoxyphenyl)piperazino]sulfonylphenyl]oxazole | 2-cyclopropyl-5-[4-[[4-(3-methoxyphenyl)-1-piperazinyl]sulfonyl]phenyl]oxazole | MLS001095642 | SMR000631514 | cid_16027935

Type

Small organic molecule

Emp. Form.

C23H25N3O4S

Mol. Mass.

439.527

SMILES

COc1cccc(c1)N1CCN(CC1)S(=O)(=O)c1ccc(cc1)-c1cnc(o1)C1CC1

Structure