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TargetPhotoreceptor-specific nuclear receptor
LigandBDBM66180
Substrate/Competitorn/a
Meas. Tech.TR-FRET-based biochemical high throughput dose response assay for agonists of nuclear receptor subfamily 2, group E, member 3 (NR2E3)
IC50 1903±n/a nM
Citation PubChem, PC TR-FRET-based biochemical high throughput dose response assay for agonists of nuclear receptor subfamily 2, group E, member 3 (NR2E3) PubChem Bioassay(2010)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Photoreceptor-specific nuclear receptor
Name:Photoreceptor-specific nuclear receptor
Synonyms:NR2E3 | NR2E3_HUMAN | PNR | RNR | photoreceptor-specific nuclear receptor
Type:PROTEIN
Mol. Mass.:44699.83
Organism:Homo sapiens (Human)
Description:ChEMBL_401901
Residue:410
Sequence:
METRPTALMSSTVAAAAPAAGAASRKESPGRWGLGEDPTGVSPSLQCRVCGDSSSGKHYG
IYACNGCSGFFKRSVRRRLIYRCQVGAGMCPVDKAHRNQCQACRLKKCLQAGMNQDAVQN
ERQPRSTAQVHLDSMESNTESRPESLVAPPAPAGRSPRGPTPMSAARALGHHFMASLITA
ETCAKLEPEDADENIDVTSNDPEFPSSPYSSSSPCGLDSIHETSARLLFMAVKWAKNLPV
FSSLPFRDQVILLEEAWSELFLLGAIQWSLPLDSCPLLAPPEASAAGGAQGRLTLASMET
RVLQETISRFRALAVDPTEFACMKALVLFKPETRGLKDPEHVEALQDQSQVMLSQHSKAH
HPSQPVRFGKLLLLLPSLRFITAERIELLFFRKTIGNTPMEKLLCDMFKN
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  Blast E-value cutoff:
BDBM66180
n/a
NameBDBM66180
Synonyms:5-Isopropyl-10-thioxo-1,2,3,4,10,11-hexahydro-9H-7-thia-6,9,11-triaza-benzo[c]fluoren-8-one | MLS000778188 | SMR000414964 | cid_929935
TypeSmall organic molecule
Emp. Form.C16H17N3OS2
Mol. Mass.331.456
SMILESCC(C)c1nc2sc3c([nH]c(=S)[nH]c3=O)c2c2CCCCc12
Structure
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