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TargetPhotoreceptor-specific nuclear receptor
LigandBDBM66193
Substrate/Competitorn/a
Meas. Tech.TR-FRET-based biochemical high throughput dose response assay for agonists of nuclear receptor subfamily 2, group E, member 3 (NR2E3)
IC50 220.17±n/a nM
Citation PubChem, PC TR-FRET-based biochemical high throughput dose response assay for agonists of nuclear receptor subfamily 2, group E, member 3 (NR2E3) PubChem Bioassay(2010)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Photoreceptor-specific nuclear receptor
Name:Photoreceptor-specific nuclear receptor
Synonyms:NR2E3 | NR2E3_HUMAN | PNR | RNR | photoreceptor-specific nuclear receptor
Type:PROTEIN
Mol. Mass.:44699.83
Organism:Homo sapiens (Human)
Description:ChEMBL_401901
Residue:410
Sequence:
METRPTALMSSTVAAAAPAAGAASRKESPGRWGLGEDPTGVSPSLQCRVCGDSSSGKHYG
IYACNGCSGFFKRSVRRRLIYRCQVGAGMCPVDKAHRNQCQACRLKKCLQAGMNQDAVQN
ERQPRSTAQVHLDSMESNTESRPESLVAPPAPAGRSPRGPTPMSAARALGHHFMASLITA
ETCAKLEPEDADENIDVTSNDPEFPSSPYSSSSPCGLDSIHETSARLLFMAVKWAKNLPV
FSSLPFRDQVILLEEAWSELFLLGAIQWSLPLDSCPLLAPPEASAAGGAQGRLTLASMET
RVLQETISRFRALAVDPTEFACMKALVLFKPETRGLKDPEHVEALQDQSQVMLSQHSKAH
HPSQPVRFGKLLLLLPSLRFITAERIELLFFRKTIGNTPMEKLLCDMFKN
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  Blast E-value cutoff:
BDBM66193
n/a
NameBDBM66193
Synonyms:7-(4-methoxyphenyl)-5-phenyl-4-pyrido[2,3-d]pyrimidinamine | 7-(4-methoxyphenyl)-5-phenyl-pyrido[2,3-d]pyrimidin-4-amine | 7-(4-methoxyphenyl)-5-phenylpyrido[2,3-d]pyrimidin-4-amine | MLS001181933 | SMR000567698 | [7-(4-methoxyphenyl)-5-phenyl-pyrido[2,3-d]pyrimidin-4-yl]amine | cid_2817025
TypeSmall organic molecule
Emp. Form.C20H16N4O
Mol. Mass.328.3672
SMILESCOc1ccc(cc1)-c1cc(-c2ccccc2)c2c(N)ncnc2n1
Structure
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