| Reaction Details |
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 | Report a problem with these data |
| Target | Serine/threonine-protein kinase 33 |
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| Ligand | BDBM24713 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Luminescence Cell-Free Homogenous Dose Retest to Identify Inhibitors of Serine/Threonine Kinase 33 Activity |
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| EC50 | 60970±n/a nM |
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| Citation |  PubChem, PC Luminescence Cell-Free Homogenous Dose Retest to Identify Inhibitors of Serine/Threonine Kinase 33 Activity PubChem Bioassay(2010)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| Serine/threonine-protein kinase 33 |
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| Name: | Serine/threonine-protein kinase 33 |
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| Synonyms: | STK33 | STK33_HUMAN | Serine/threonine-protein kinase 33 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 57833.21 |
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| Organism: | Homo sapiens (Human) |
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| Description: | gi_23943882 |
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| Residue: | 514 |
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| Sequence: | MADSGLDKKSTKCPDCSSASQKDVLCVCSSKTRVPPVLVVEMSQTSSIGSAESLISLERK
KEKNINRDITSRKDLPSRTSNVERKASQQQWGRGNFTEGKVPHIRIENGAAIEEIYTFGR
ILGKGSFGIVIEATDKETETKWAIKKVNKEKAGSSAVKLLEREVNILKSVKHEHIIHLEQ
VFETPKKMYLVMELCEDGELKEILDRKGHFSENETRWIIQSLASAIAYLHNNDIVHRDLK
LENIMVKSSLIDDNNEINLNIKVTDFGLAVKKQSRSEAMLQATCGTPIYMAPEVISAHDY
SQQCDIWSIGVVMYMLLRGEPPFLASSEEKLFELIRKGELHFENAVWNSISDCAKSVLKQ
LMKVDPAHRITAKELLDNQWLTGNKLSSVRPTNVLEMMKEWKNNPESVEENTTEEKNKPS
TEEKLKSYQPWGNVPDANYTSDEEEEKQSTAYEKQFPATSKDNFDMCSSSFTSSKLLPAE
IKGEMEKTPVTPSQGTATKYPAKSGALSRTKKKL
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| BDBM24713 |
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| n/a |
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| Name | BDBM24713 |
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| Synonyms: | 1,2,4,5-tetrahydropyrazolo[3,4-a]carbazole | 3,4,16-triazatetracyclo[7.7.0.0^{2,6}.0^{10,15}]hexadeca-1(9),2,5,10,12,14-hexaene | Tetrahydropyrazolo[3,4-a]carbazole, 19 |
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| Type | Small organic molecule |
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| Emp. Form. | C13H11N3 |
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| Mol. Mass. | 209.2465 |
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| SMILES | C1Cc2c([nH]c3ccccc23)-c2n[nH]cc12 |
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| Structure | 
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