| Reaction Details |
|---|
 | Report a problem with these data |
| Target | G-protein coupled receptor 35 |
|---|
| Ligand | BDBM68293 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | SAR analysis of Antagonists of the GPR35 Receptor using an Image-Based Assay - Set 4 |
|---|
| IC50 | >32000±n/a nM |
|---|
| Citation |  PubChem, PC SAR analysis of Antagonists of the GPR35 Receptor using an Image-Based Assay - Set 4 PubChem Bioassay(2010)[AID] |
|---|
| More Info.: | Get all data from this article, Solution Info, Assay Method |
|---|
| |
| G-protein coupled receptor 35 |
|---|
| Name: | G-protein coupled receptor 35 |
|---|
| Synonyms: | G protein-coupled receptor 35 | GPR35 | GPR35_HUMAN |
|---|
| Type: | Enzyme Catalytic Domain |
|---|
| Mol. Mass.: | 34085.57 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | gi_33695097 |
|---|
| Residue: | 309 |
|---|
| Sequence: | MNGTYNTCGSSDLTWPPAIKLGFYAYLGVLLVLGLLLNSLALWVFCCRMQQWTETRIYMT
NLAVADLCLLCTLPFVLHSLRDTSDTPLCQLSQGIYLTNRYMSISLVTAIAVDRYVAVRH
PLRARGLRSPRQAAAVCAVLWVLVIGSLVARWLLGIQEGGFCFRSTRHNFNSMAFPLLGF
YLPLAVVVFCSLKVVTALAQRPPTDVGQAEATRKAARMVWANLLVFVVCFLPLHVGLTVR
LAVGWNACALLETIRRALYITSKLSDANCCLDAICYYYMAKEFQEASALAVAPSAKAHKS
QDSLCVTLA
|
|
|
|---|
| BDBM68293 |
|---|
| n/a |
|---|
| Name | BDBM68293 |
|---|
| Synonyms: | 3-[4-(2,3-dimethylphenyl)piperazin-1-yl]carbonyl-N,N-dimethyl-benzenesulfonamide | 3-[4-(2,3-dimethylphenyl)piperazine-1-carbonyl]-N,N-dimethyl-benzenesulfonamide | 3-[4-(2,3-dimethylphenyl)piperazine-1-carbonyl]-N,N-dimethylbenzenesulfonamide | 3-[[4-(2,3-dimethylphenyl)-1-piperazinyl]-oxomethyl]-N,N-dimethylbenzenesulfonamide | MLS-0435526.0001 | cid_2090194 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C21H27N3O3S |
|---|
| Mol. Mass. | 401.522 |
|---|
| SMILES | CN(C)S(=O)(=O)c1cccc(c1)C(=O)N1CCN(CC1)c1cccc(C)c1C |
|---|
| Structure | 
|
|---|
Search and Browse
