Ki Summary

Reaction Details

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Target

Krueppel-like factor 5

Ligand

BDBM70197

Substrate/Competitor

n/a

Meas. Tech.

Late stage results from the probe development effort to identify inhibitors of kruppel-like factor 5 (KLF5): luminescence-based cell-based dose response assay for inhibitors of KLF5 (Round 1)

IC50

>39841±n/a nM

Citation

PubChem, PC Late stage results from the probe development effort to identify inhibitors of kruppel-like factor 5 (KLF5): luminescence-based cell-based dose response assay for inhibitors of KLF5 (Round 1) PubChem Bioassay(2010)[AID]

More Info.:

Get all data from this article, Solution Info, Assay Method

Krueppel-like factor 5

Name:

Krueppel-like factor 5

Synonyms:

Type:

Enzyme Catalytic Domain

Mol. Mass.:

50808.71

Organism:

Homo sapiens (Human)

Description:

Q13887

Residue:

457

Sequence:

MATRVLSMSARLGPVPQPPAPQDEPVFAQLKPVLGAANPARDAALFPGEELKHAHHRPQA
QPAPAQAPQPAQPPATGPRLPPEDLVQTRCEMEKYLTPQLPPVPIIPEHKKYRRDSASVV
DQFFTDTEGLPYSINMNVFLPDITHLRTGLYKSQRPCVTHIKTEPVAIFSHQSETTAPPP
APTQALPEFTSIFSSHQTAAPEVNNIFIKQELPTPDLHLSVPTQQGHLYQLLNTPDLDMP
SSTNQTAAMDTLNVSMSAAMAGLNTHTSAVPQTAVKQFQGMPPCTYTMPSQFLPQQATYF
PPSPPSSEPGSPDRQAEMLQNLTPPPSYAATIASKLAIHNPNLPTTLPVNSQNIQPVRYN
RRSNPDLEKRRIHYCDYPGCTKVYTKSSHLKAHLRTHTGEKPYKCTWEGCDWRFARSDEL
TRHYRKHTGAKPFQCGVCNRSFSRSDHLALHMKRHQN

BDBM70197

n/a

Name

BDBM70197

Synonyms:

N-[2-(3-chlorophenyl)-5-benzotriazolyl]-2-phenoxyacetamide | N-[2-(3-chlorophenyl)benzotriazol-5-yl]-2-phenoxy-acetamide | N-[2-(3-chlorophenyl)benzotriazol-5-yl]-2-phenoxy-ethanamide | N-[2-(3-chlorophenyl)benzotriazol-5-yl]-2-phenoxyacetamide | SR-01000419352 | SR-01000419352-2 | cid_1112727

Type

Small organic molecule

Emp. Form.

C20H15ClN4O2

Mol. Mass.

378.812

SMILES

Clc1cccc(c1)-n1nc2ccc(NC(=O)COc3ccccc3)cc2n1

Structure