Ki Summary

Reaction Details

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Target

Krueppel-like factor 5

Ligand

BDBM70200

Substrate/Competitor

n/a

Meas. Tech.

Late stage results from the probe development effort to identify inhibitors of kruppel-like factor 5 (KLF5): luminescence-based cell-based dose response assay for inhibitors of KLF5 (Round 1)

IC50

>39841±n/a nM

Citation

PubChem, PC Late stage results from the probe development effort to identify inhibitors of kruppel-like factor 5 (KLF5): luminescence-based cell-based dose response assay for inhibitors of KLF5 (Round 1) PubChem Bioassay(2010)[AID]

More Info.:

Get all data from this article, Solution Info, Assay Method

Krueppel-like factor 5

Name:

Krueppel-like factor 5

Synonyms:

Type:

Enzyme Catalytic Domain

Mol. Mass.:

50808.71

Organism:

Homo sapiens (Human)

Description:

Q13887

Residue:

457

Sequence:

MATRVLSMSARLGPVPQPPAPQDEPVFAQLKPVLGAANPARDAALFPGEELKHAHHRPQA
QPAPAQAPQPAQPPATGPRLPPEDLVQTRCEMEKYLTPQLPPVPIIPEHKKYRRDSASVV
DQFFTDTEGLPYSINMNVFLPDITHLRTGLYKSQRPCVTHIKTEPVAIFSHQSETTAPPP
APTQALPEFTSIFSSHQTAAPEVNNIFIKQELPTPDLHLSVPTQQGHLYQLLNTPDLDMP
SSTNQTAAMDTLNVSMSAAMAGLNTHTSAVPQTAVKQFQGMPPCTYTMPSQFLPQQATYF
PPSPPSSEPGSPDRQAEMLQNLTPPPSYAATIASKLAIHNPNLPTTLPVNSQNIQPVRYN
RRSNPDLEKRRIHYCDYPGCTKVYTKSSHLKAHLRTHTGEKPYKCTWEGCDWRFARSDEL
TRHYRKHTGAKPFQCGVCNRSFSRSDHLALHMKRHQN

BDBM70200

n/a

Name

BDBM70200

Synonyms:

N-[2-(4-methoxyphenyl)-5-benzotriazolyl]-2,2-dimethylpropanamide | N-[2-(4-methoxyphenyl)benzotriazol-5-yl]-2,2-dimethyl-propanamide | N-[2-(4-methoxyphenyl)benzotriazol-5-yl]-2,2-dimethyl-propionamide | N-[2-(4-methoxyphenyl)benzotriazol-5-yl]-2,2-dimethylpropanamide | SR-03000001316 | SR-03000001316-1 | cid_17027238

Type

Small organic molecule

Emp. Form.

C18H20N4O2

Mol. Mass.

324.377

SMILES

COc1ccc(cc1)-n1nc2ccc(NC(=O)C(C)(C)C)cc2n1

Structure