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TargetKruppel-like factor 5
LigandBDBM70203
Substrate/Competitorn/a
Meas. Tech.Late stage results from the probe development effort to identify inhibitors of kruppel-like factor 5 (KLF5): luminescence-based cell-based dose response assay for inhibitors of KLF5 (Round 1)
IC50 26285±n/a nM
Citation PubChem PC Late stage results from the probe development effort to identify inhibitors of kruppel-like factor 5 (KLF5): luminescence-based cell-based dose response assay for inhibitors of KLF5 (Round 1) PubChem Bioassay (2010)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Kruppel-like factor 5
Name:Kruppel-like factor 5
Synonyms:n/a
Type:Enzyme Catalytic Domain
Mol. Mass.:50808.71
Organism:Homo sapiens (Human)
Description:Q13887
Residue:457
Sequence:
MATRVLSMSARLGPVPQPPAPQDEPVFAQLKPVLGAANPARDAALFPGEELKHAHHRPQA
QPAPAQAPQPAQPPATGPRLPPEDLVQTRCEMEKYLTPQLPPVPIIPEHKKYRRDSASVV
DQFFTDTEGLPYSINMNVFLPDITHLRTGLYKSQRPCVTHIKTEPVAIFSHQSETTAPPP
APTQALPEFTSIFSSHQTAAPEVNNIFIKQELPTPDLHLSVPTQQGHLYQLLNTPDLDMP
SSTNQTAAMDTLNVSMSAAMAGLNTHTSAVPQTAVKQFQGMPPCTYTMPSQFLPQQATYF
PPSPPSSEPGSPDRQAEMLQNLTPPPSYAATIASKLAIHNPNLPTTLPVNSQNIQPVRYN
RRSNPDLEKRRIHYCDYPGCTKVYTKSSHLKAHLRTHTGEKPYKCTWEGCDWRFARSDEL
TRHYRKHTGAKPFQCGVCNRSFSRSDHLALHMKRHQN
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  Blast E-value cutoff:
BDBM70203
n/a
NameBDBM70203
Synonyms:N-[2-(4-chlorophenyl)-5-benzotriazolyl]-2-methylpropanamide | N-[2-(4-chlorophenyl)benzotriazol-5-yl]-2-methyl-propanamide | N-[2-(4-chlorophenyl)benzotriazol-5-yl]-2-methyl-propionamide | N-[2-(4-chlorophenyl)benzotriazol-5-yl]-2-methylpropanamide | SR-03000001320 | SR-03000001320-1 | cid_881898
TypeSmall organic molecule
Emp. Form.C16H15ClN4O
Mol. Mass.314.77
SMILESCC(C)C(=O)Nc1ccc2nn(nc2c1)-c1ccc(Cl)cc1
Structure
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