Ki Summary

Reaction Details

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Target

Krueppel-like factor 5

Ligand

BDBM70204

Substrate/Competitor

n/a

Meas. Tech.

Late stage results from the probe development effort to identify inhibitors of kruppel-like factor 5 (KLF5): luminescence-based cell-based dose response assay for inhibitors of KLF5 (Round 1)

IC50

>39841±n/a nM

Citation

PubChem, PC Late stage results from the probe development effort to identify inhibitors of kruppel-like factor 5 (KLF5): luminescence-based cell-based dose response assay for inhibitors of KLF5 (Round 1) PubChem Bioassay(2010)[AID]

More Info.:

Get all data from this article, Solution Info, Assay Method

Krueppel-like factor 5

Name:

Krueppel-like factor 5

Synonyms:

Type:

Enzyme Catalytic Domain

Mol. Mass.:

50808.71

Organism:

Homo sapiens (Human)

Description:

Q13887

Residue:

457

Sequence:

MATRVLSMSARLGPVPQPPAPQDEPVFAQLKPVLGAANPARDAALFPGEELKHAHHRPQA
QPAPAQAPQPAQPPATGPRLPPEDLVQTRCEMEKYLTPQLPPVPIIPEHKKYRRDSASVV
DQFFTDTEGLPYSINMNVFLPDITHLRTGLYKSQRPCVTHIKTEPVAIFSHQSETTAPPP
APTQALPEFTSIFSSHQTAAPEVNNIFIKQELPTPDLHLSVPTQQGHLYQLLNTPDLDMP
SSTNQTAAMDTLNVSMSAAMAGLNTHTSAVPQTAVKQFQGMPPCTYTMPSQFLPQQATYF
PPSPPSSEPGSPDRQAEMLQNLTPPPSYAATIASKLAIHNPNLPTTLPVNSQNIQPVRYN
RRSNPDLEKRRIHYCDYPGCTKVYTKSSHLKAHLRTHTGEKPYKCTWEGCDWRFARSDEL
TRHYRKHTGAKPFQCGVCNRSFSRSDHLALHMKRHQN

BDBM70204

n/a

Name

BDBM70204

Synonyms:

N-[6-chloranyl-2-(4-methylphenyl)benzotriazol-5-yl]pyridine-3-carboxamide | N-[6-chloro-2-(4-methylphenyl)-5-benzotriazolyl]-3-pyridinecarboxamide | N-[6-chloro-2-(4-methylphenyl)benzotriazol-5-yl]pyridine-3-carboxamide | N-[6-chloro-2-(p-tolyl)benzotriazol-5-yl]nicotinamide | SR-03000001321 | SR-03000001321-1 | cid_1071621

Type

Small organic molecule

Emp. Form.

C19H14ClN5O

Mol. Mass.

363.8

SMILES

Cc1ccc(cc1)-n1nc2cc(Cl)c(NC(=O)c3cccnc3)cc2n1

Structure