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TargetKruppel-like factor 5
LigandBDBM70204
Substrate/Competitorn/a
Meas. Tech.Late stage results from the probe development effort to identify inhibitors of kruppel-like factor 5 (KLF5): luminescence-based cell-based dose response assay for inhibitors of KLF5 (Round 1)
IC50>39841±n/a nM
Citation PubChem PC Late stage results from the probe development effort to identify inhibitors of kruppel-like factor 5 (KLF5): luminescence-based cell-based dose response assay for inhibitors of KLF5 (Round 1) PubChem Bioassay (2010)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Kruppel-like factor 5
Name:Kruppel-like factor 5
Synonyms:n/a
Type:Enzyme Catalytic Domain
Mol. Mass.:50808.71
Organism:Homo sapiens (Human)
Description:Q13887
Residue:457
Sequence:
MATRVLSMSARLGPVPQPPAPQDEPVFAQLKPVLGAANPARDAALFPGEELKHAHHRPQA
QPAPAQAPQPAQPPATGPRLPPEDLVQTRCEMEKYLTPQLPPVPIIPEHKKYRRDSASVV
DQFFTDTEGLPYSINMNVFLPDITHLRTGLYKSQRPCVTHIKTEPVAIFSHQSETTAPPP
APTQALPEFTSIFSSHQTAAPEVNNIFIKQELPTPDLHLSVPTQQGHLYQLLNTPDLDMP
SSTNQTAAMDTLNVSMSAAMAGLNTHTSAVPQTAVKQFQGMPPCTYTMPSQFLPQQATYF
PPSPPSSEPGSPDRQAEMLQNLTPPPSYAATIASKLAIHNPNLPTTLPVNSQNIQPVRYN
RRSNPDLEKRRIHYCDYPGCTKVYTKSSHLKAHLRTHTGEKPYKCTWEGCDWRFARSDEL
TRHYRKHTGAKPFQCGVCNRSFSRSDHLALHMKRHQN
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  Blast E-value cutoff:
BDBM70204
n/a
NameBDBM70204
Synonyms:N-[6-chloranyl-2-(4-methylphenyl)benzotriazol-5-yl]pyridine-3-carboxamide | N-[6-chloro-2-(4-methylphenyl)-5-benzotriazolyl]-3-pyridinecarboxamide | N-[6-chloro-2-(4-methylphenyl)benzotriazol-5-yl]pyridine-3-carboxamide | N-[6-chloro-2-(p-tolyl)benzotriazol-5-yl]nicotinamide | SR-03000001321 | SR-03000001321-1 | cid_1071621
TypeSmall organic molecule
Emp. Form.C19H14ClN5O
Mol. Mass.363.8
SMILESCc1ccc(cc1)-n1nc2cc(Cl)c(NC(=O)c3cccnc3)cc2n1
Structure
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