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TargetKruppel-like factor 5
LigandBDBM70225
Substrate/Competitorn/a
Meas. Tech.Late stage results from the probe development effort to identify inhibitors of kruppel-like factor 5 (KLF5): luminescence-based cell-based dose response assay for inhibitors of KLF5 (Round 1)
IC50 7965±n/a nM
Citation PubChem PC Late stage results from the probe development effort to identify inhibitors of kruppel-like factor 5 (KLF5): luminescence-based cell-based dose response assay for inhibitors of KLF5 (Round 1) PubChem Bioassay (2010)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Kruppel-like factor 5
Name:Kruppel-like factor 5
Synonyms:n/a
Type:Enzyme Catalytic Domain
Mol. Mass.:50808.71
Organism:Homo sapiens (Human)
Description:Q13887
Residue:457
Sequence:
MATRVLSMSARLGPVPQPPAPQDEPVFAQLKPVLGAANPARDAALFPGEELKHAHHRPQA
QPAPAQAPQPAQPPATGPRLPPEDLVQTRCEMEKYLTPQLPPVPIIPEHKKYRRDSASVV
DQFFTDTEGLPYSINMNVFLPDITHLRTGLYKSQRPCVTHIKTEPVAIFSHQSETTAPPP
APTQALPEFTSIFSSHQTAAPEVNNIFIKQELPTPDLHLSVPTQQGHLYQLLNTPDLDMP
SSTNQTAAMDTLNVSMSAAMAGLNTHTSAVPQTAVKQFQGMPPCTYTMPSQFLPQQATYF
PPSPPSSEPGSPDRQAEMLQNLTPPPSYAATIASKLAIHNPNLPTTLPVNSQNIQPVRYN
RRSNPDLEKRRIHYCDYPGCTKVYTKSSHLKAHLRTHTGEKPYKCTWEGCDWRFARSDEL
TRHYRKHTGAKPFQCGVCNRSFSRSDHLALHMKRHQN
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  Blast E-value cutoff:
BDBM70225
n/a
NameBDBM70225
Synonyms:N-(6-chloranyl-2-phenyl-benzotriazol-5-yl)-2-phenyl-ethanamide | N-(6-chloro-2-phenyl-5-benzotriazolyl)-2-phenylacetamide | N-(6-chloro-2-phenyl-benzotriazol-5-yl)-2-phenyl-acetamide | N-(6-chloro-2-phenylbenzotriazol-5-yl)-2-phenylacetamide | SR-03000001356 | SR-03000001356-1 | cid_1305859
TypeSmall organic molecule
Emp. Form.C20H15ClN4O
Mol. Mass.362.812
SMILESClc1cc2nn(nc2cc1NC(=O)Cc1ccccc1)-c1ccccc1
Structure
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