| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Protein LANA1 |
|---|
| Ligand | BDBM74282 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | Fluorescence Polarization Cell-Free Homogeneous Dose Retest to Confirm Inhibitors of the LANA Histone H2A/H2B Interaction |
|---|
| EC50 | >75000±n/a nM |
|---|
| Citation |  PubChem, PC Fluorescence Polarization Cell-Free Homogeneous Dose Retest to Confirm Inhibitors of the LANA Histone H2A/H2B Interaction PubChem Bioassay(2010)[AID] |
|---|
| More Info.: | Get all data from this article, Solution Info, Assay Method |
|---|
| |
| Protein LANA1 |
|---|
| Name: | Protein LANA1 |
|---|
| Synonyms: | LANA | LANA1 | LANA1_HHV8P |
|---|
| Type: | Enzyme Catalytic Domain |
|---|
| Mol. Mass.: | 131093.36 |
|---|
| Organism: | Human herpesvirus 8 |
|---|
| Description: | Q9QR71 |
|---|
| Residue: | 1129 |
|---|
| Sequence: | MAPPGMRLRSGRSTGAPLTRGSCRKRNRSPERCDLGDDLHLQPRRKHVADSVDGRECGPH
TLPIPGSPTVFTSGLPAFVSSPTLPVAPIPSPAPATPLPPPALLPPVTTSSSPIPPSHPV
SPGTTDTHSPSPALPPTQSPESSQRPPLSSPTGRPDSSTPMRPPPSQQTTPPHSPTTPPP
EPPSKSSPDSLAPSTLRSLRKRRLSSPQGPSTLNPICQSPPVSPPRCDFANRSVYPPWAT
ESPIYVGSSSDGDTPPRQPPTSPISIGSSSPSEGSWGDDTAMLVLLAEIAEEASKNEKEC
SENNQAGEDNGDNEISKESQVDKDDNDNKDDEEEQETDEEDEEDDEEDDEEDDEEDDEED
DEEDDEEDDEEEDEEEDEEEDEEEDEEEEEDEEDDDDEDNEDEEDDEEEDKKEDEEDGGD
GNKTLSIQSSQQQQEPQQQEPQQQEPQQQEPQQQEPQQQEPQQQEPQQQEPQQREPQQRE
PQQREPQQREPQQREPQQREPQQREPQQREPQQREPQQREPQQREPQQREPQQQEPQQQE
PQQQEPQQQEPQQQEPQQQEPQQQEPQQQEPQQQEPQQQEPQQQEPQQQEPQQQDEQQQD
EQQQDEQQQDEQQQDEQQQDEQQQDEQQQDEQEQQDEQQQDEQQQQDEQEQQEEQEQQEE
QQQDEQQQDEQQQDEQQQDEQEQQDEQQQDEQQQQDEQEQQEEQEQQEEQEQQEEQEQQE
EQEQELEEQEQELEEQEQELEEQEQELEEQEQELEEQEQELEEQEQELEEQEQELEEQEQ
ELEEQEQELEEQEQELEEQEQELEEQEQELEEQEQELEEQEQEQELEEVEEQEQEQEEQE
LEEVEEQEQEQEEQEEQELEEVEEQEEQELEEVEEQEEQELEEVEEQEQQGVEQQEQETV
EEPIILHGSSSEDEMEVDYPVVSTHEQIASSPPGDNTPDDDPQPGPSREYRYVLRTSPPH
RPGVRMRRVPVTHPKKPHPRYQQPPVPYRQIDDCPAKARPQHIFYRRFLGKDGRRDPKCQ
WKFAVIFWGNDPYGLKKLSQAFQFGGVKAGPVSCLPHPGPDQSPITYCVYVYCQNKDTSK
KVQMARLAWEASHPLAGNLQSSIVKFKKPLPLTQPGENQGPGDSPQEMT
|
|
|
|---|
| BDBM74282 |
|---|
| n/a |
|---|
| Name | BDBM74282 |
|---|
| Synonyms: | MLS002182844 | N-[2-(dimethylamino)-2-phenyl-ethyl]-2-methyl-5-(m-tolylsulfamoyl)benzamide | N-[2-(dimethylamino)-2-phenyl-ethyl]-2-methyl-5-[(3-methylphenyl)sulfamoyl]benzamide | N-[2-(dimethylamino)-2-phenylethyl]-2-methyl-5-[(3-methylphenyl)sulfamoyl]benzamide | SMR001271874 | cid_25161888 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C25H29N3O3S |
|---|
| Mol. Mass. | 451.581 |
|---|
| SMILES | CN(C)C(CNC(=O)c1cc(ccc1C)S(=O)(=O)Nc1cccc(C)c1)c1ccccc1 |
|---|
| Structure | 
|
|---|
Search and Browse
