| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Protein LANA1 |
|---|
| Ligand | BDBM74299 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | Fluorescence Polarization Cell-Free Homogeneous Dose Retest to Confirm Inhibitors of the LANA Histone H2A/H2B Interaction |
|---|
| EC50 | >75000±n/a nM |
|---|
| Citation |  PubChem, PC Fluorescence Polarization Cell-Free Homogeneous Dose Retest to Confirm Inhibitors of the LANA Histone H2A/H2B Interaction PubChem Bioassay(2010)[AID] |
|---|
| More Info.: | Get all data from this article, Solution Info, Assay Method |
|---|
| |
| Protein LANA1 |
|---|
| Name: | Protein LANA1 |
|---|
| Synonyms: | LANA | LANA1 | LANA1_HHV8P |
|---|
| Type: | Enzyme Catalytic Domain |
|---|
| Mol. Mass.: | 131093.36 |
|---|
| Organism: | Human herpesvirus 8 |
|---|
| Description: | Q9QR71 |
|---|
| Residue: | 1129 |
|---|
| Sequence: | MAPPGMRLRSGRSTGAPLTRGSCRKRNRSPERCDLGDDLHLQPRRKHVADSVDGRECGPH
TLPIPGSPTVFTSGLPAFVSSPTLPVAPIPSPAPATPLPPPALLPPVTTSSSPIPPSHPV
SPGTTDTHSPSPALPPTQSPESSQRPPLSSPTGRPDSSTPMRPPPSQQTTPPHSPTTPPP
EPPSKSSPDSLAPSTLRSLRKRRLSSPQGPSTLNPICQSPPVSPPRCDFANRSVYPPWAT
ESPIYVGSSSDGDTPPRQPPTSPISIGSSSPSEGSWGDDTAMLVLLAEIAEEASKNEKEC
SENNQAGEDNGDNEISKESQVDKDDNDNKDDEEEQETDEEDEEDDEEDDEEDDEEDDEED
DEEDDEEDDEEEDEEEDEEEDEEEDEEEEEDEEDDDDEDNEDEEDDEEEDKKEDEEDGGD
GNKTLSIQSSQQQQEPQQQEPQQQEPQQQEPQQQEPQQQEPQQQEPQQQEPQQREPQQRE
PQQREPQQREPQQREPQQREPQQREPQQREPQQREPQQREPQQREPQQREPQQQEPQQQE
PQQQEPQQQEPQQQEPQQQEPQQQEPQQQEPQQQEPQQQEPQQQEPQQQEPQQQDEQQQD
EQQQDEQQQDEQQQDEQQQDEQQQDEQQQDEQEQQDEQQQDEQQQQDEQEQQEEQEQQEE
QQQDEQQQDEQQQDEQQQDEQEQQDEQQQDEQQQQDEQEQQEEQEQQEEQEQQEEQEQQE
EQEQELEEQEQELEEQEQELEEQEQELEEQEQELEEQEQELEEQEQELEEQEQELEEQEQ
ELEEQEQELEEQEQELEEQEQELEEQEQELEEQEQELEEQEQEQELEEVEEQEQEQEEQE
LEEVEEQEQEQEEQEEQELEEVEEQEEQELEEVEEQEEQELEEVEEQEQQGVEQQEQETV
EEPIILHGSSSEDEMEVDYPVVSTHEQIASSPPGDNTPDDDPQPGPSREYRYVLRTSPPH
RPGVRMRRVPVTHPKKPHPRYQQPPVPYRQIDDCPAKARPQHIFYRRFLGKDGRRDPKCQ
WKFAVIFWGNDPYGLKKLSQAFQFGGVKAGPVSCLPHPGPDQSPITYCVYVYCQNKDTSK
KVQMARLAWEASHPLAGNLQSSIVKFKKPLPLTQPGENQGPGDSPQEMT
|
|
|
|---|
| BDBM74299 |
|---|
| n/a |
|---|
| Name | BDBM74299 |
|---|
| Synonyms: | MLS002182290 | N-[3-(1-azepanylsulfonyl)-4-methylphenyl]-2-(3-oxo-1H-isobenzofuran-1-yl)acetamide | N-[3-(azepan-1-ylsulfonyl)-4-methyl-phenyl]-2-(3-oxidanylidene-1H-2-benzofuran-1-yl)ethanamide | N-[3-(azepan-1-ylsulfonyl)-4-methyl-phenyl]-2-phthalidyl-acetamide | N-[3-(azepan-1-ylsulfonyl)-4-methylphenyl]-2-(3-oxo-1H-2-benzofuran-1-yl)acetamide | SMR001271320 | cid_25162545 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C23H26N2O5S |
|---|
| Mol. Mass. | 442.528 |
|---|
| SMILES | Cc1ccc(NC(=O)CC2OC(=O)c3ccccc23)cc1S(=O)(=O)N1CCCCCC1 |
|---|
| Structure | 
|
|---|
Search and Browse
