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TargetTyrosine-protein phosphatase non-receptor type 7
LigandBDBM74450
Substrate/Competitorn/a
Meas. Tech.Dose Response confirmation of HTS hits from an HePTP Fluorescent Assay using OMFP substrate - Set 2
IC50>79400±0 nM
Citation PubChem, PC Dose Response confirmation of HTS hits from an HePTP Fluorescent Assay using OMFP substrate - Set 2 PubChem Bioassay(2010)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Tyrosine-protein phosphatase non-receptor type 7
Name:Tyrosine-protein phosphatase non-receptor type 7
Synonyms:He-PTP | Hematopoietic protein-tyrosine phosphatase | Hematopoietic protein-tyrosine phosphatase (HEPTP) | PTN7_HUMAN | PTPN7 | Protein-tyrosine phosphatase LC-PTP | Tyrosine-protein phosphatase non-receptor type 7 | Tyrosine-protein phosphatase non-receptor type 7 (HEPTP)
Type:Protein
Mol. Mass.:40530.79
Organism:Homo sapiens (Human)
Description:P35236
Residue:360
Sequence:
MVQAHGGRSRAQPLTLSLGAAMTQPPPEKTPAKKHVRLQERRGSNVALMLDVRSLGAVEP
ICSVNTPREVTLHFLRTAGHPLTRWALQRQPPSPKQLEEEFLKIPSNFVSPEDLDIPGHA
SKDRYKTILPNPQSRVCLGRAQSQEDGDYINANYIRGYDGKEKVYIATQGPMPNTVSDFW
EMVWQEEVSLIVMLTQLREGKEKCVHYWPTEEETYGPFQIRIQDMKECPEYTVRQLTIQY
QEERRSVKHILFSAWPDHQTPESAGPLLRLVAEVEESPETAAHPGPIVVHCSAGIGRTGC
FIATRIGCQQLKARGEVDILGIVCQLRLDRGGMIQTAEQYQFLHHTLALYAGQLPEEPSP
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  Blast E-value cutoff:
BDBM74450
n/a
NameBDBM74450
Synonyms:3-[2-(2,3,5,6-tetrafluoro-4-methylol-anilino)ethylamino]cyclohex-2-en-1-one | 3-[2-[2,3,5,6-tetrafluoro-4-(hydroxymethyl)anilino]ethylamino]-1-cyclohex-2-enone | 3-[2-[2,3,5,6-tetrafluoro-4-(hydroxymethyl)anilino]ethylamino]cyclohex-2-en-1-one | 3-[2-[[2,3,5,6-tetrakis(fluoranyl)-4-(hydroxymethyl)phenyl]amino]ethylamino]cyclohex-2-en-1-one | MLS000039349 | SMR000041400 | cid_660485
TypeSmall organic molecule
Emp. Form.C15H16F4N2O2
Mol. Mass.332.2934
SMILESOCc1c(F)c(F)c(NCCNC2=CC(=O)CCC2)c(F)c1F |t:12|
Structure
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