| Reaction Details |
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 | Report a problem with these data |
| Target | Krueppel-like factor 5 |
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| Ligand | BDBM76096 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Late stage assay provider counterscreen results from the probe development effort to identify inhibitors of kruppel-like factor 5 (KLF5) |
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| IC50 | 2246±n/a nM |
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| Citation |  PubChem, PC Late stage assay provider counterscreen results from the probe development effort to identify inhibitors of kruppel-like factor 5 (KLF5): chemiluminescence-based western blot assay for inhibitors of KLF5 protein levels PubChem Bioassay(2010)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| Krueppel-like factor 5 |
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| Name: | Krueppel-like factor 5 |
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| Synonyms: | BTEB2 | CKLF | IKLF | KLF5 | KLF5_HUMAN | Kruppel-like factor 5 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 50808.71 |
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| Organism: | Homo sapiens (Human) |
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| Description: | Q13887 |
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| Residue: | 457 |
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| Sequence: | MATRVLSMSARLGPVPQPPAPQDEPVFAQLKPVLGAANPARDAALFPGEELKHAHHRPQA
QPAPAQAPQPAQPPATGPRLPPEDLVQTRCEMEKYLTPQLPPVPIIPEHKKYRRDSASVV
DQFFTDTEGLPYSINMNVFLPDITHLRTGLYKSQRPCVTHIKTEPVAIFSHQSETTAPPP
APTQALPEFTSIFSSHQTAAPEVNNIFIKQELPTPDLHLSVPTQQGHLYQLLNTPDLDMP
SSTNQTAAMDTLNVSMSAAMAGLNTHTSAVPQTAVKQFQGMPPCTYTMPSQFLPQQATYF
PPSPPSSEPGSPDRQAEMLQNLTPPPSYAATIASKLAIHNPNLPTTLPVNSQNIQPVRYN
RRSNPDLEKRRIHYCDYPGCTKVYTKSSHLKAHLRTHTGEKPYKCTWEGCDWRFARSDEL
TRHYRKHTGAKPFQCGVCNRSFSRSDHLALHMKRHQN
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| BDBM76096 |
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| n/a |
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| Name | BDBM76096 |
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| Synonyms: | (E)-3-(3-nitrophenyl)-2-propenoic acid [2-[(1,1-dioxo-3-thiolanyl)-methylamino]-2-oxoethyl] ester | (E)-3-(3-nitrophenyl)acrylic acid [2-[(1,1-diketothiolan-3-yl)-methyl-amino]-2-keto-ethyl] ester | SR-01000765880 | SR-01000765880-2 | [2-[(1,1-dioxothiolan-3-yl)-methylamino]-2-oxoethyl] (E)-3-(3-nitrophenyl)prop-2-enoate | [2-[[1,1-bis(oxidanylidene)thiolan-3-yl]-methyl-amino]-2-oxidanylidene-ethyl] (E)-3-(3-nitrophenyl)prop-2-enoate | cid_5951923 |
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| Type | Small organic molecule |
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| Emp. Form. | C16H18N2O7S |
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| Mol. Mass. | 382.388 |
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| SMILES | CN(C1CCS(=O)(=O)C1)C(=O)COC(=O)\C=C\c1cccc(c1)[N+]([O-])=O |
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| Structure | 
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