Reaction Details |
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Target | Ubiquitin-conjugating enzyme E2 N |
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Ligand | BDBM78805 |
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Substrate/Competitor | n/a |
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Meas. Tech. | Dose Response confirmation of uHTS for the identification of UBC13 Polyubiquitin Inhibitors via a TR-FRET Assay |
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IC50 | 1677±94 nM |
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Citation | PubChem, PC Dose Response confirmation of uHTS for the identification of UBC13 Polyubiquitin Inhibitors via a TR-FRET Assay PubChem Bioassay(2011)[AID] |
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More Info.: | Get all data from this article, Solution Info, Assay Method |
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Ubiquitin-conjugating enzyme E2 N |
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Name: | Ubiquitin-conjugating enzyme E2 N |
Synonyms: | BLU | UBE2N | UBE2N_HUMAN | ubiquitin-conjugating enzyme E2 N |
Type: | PROTEIN |
Mol. Mass.: | 17137.61 |
Organism: | Homo sapiens (Human) |
Description: | EBI_101440 |
Residue: | 152 |
Sequence: | MAGLPRRIIKETQRLLAEPVPGIKAEPDESNARYFHVVIAGPQDSPFEGGTFKLELFLPE
EYPMAAPKVRFMTKIYHPNVDKLGRICLDILKDKWSPALQIRTVLLSIQALLSAPNPDDP
LANDVAEQWKTNEAQAIETARAWTRLYAMNNI
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BDBM78805 |
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n/a |
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Name | BDBM78805 |
Synonyms: | 2-amino-4-methyl-N-(3-pyridinylmethylideneamino)-5-thiazolecarboxamide | 2-amino-4-methyl-N-(3-pyridylmethyleneamino)thiazole-5-carboxamide | 2-amino-4-methyl-N-(pyridin-3-ylmethylideneamino)-1,3-thiazole-5-carboxamide | 2-azanyl-4-methyl-N-(pyridin-3-ylmethylideneamino)-1,3-thiazole-5-carboxamide | MLS000710993 | SMR000280760 | cid_772835 |
Type | Small organic molecule |
Emp. Form. | C11H11N5OS |
Mol. Mass. | 261.303 |
SMILES | Cc1nc(N)sc1C(=O)NN=Cc1cccnc1 |
Structure |
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