| Reaction Details |
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 | Report a problem with these data |
| Target | Ubiquitin-conjugating enzyme E2 N |
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| Ligand | BDBM78543 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Dose Response confirmation of uHTS for the identification of UBC13 Polyubiquitin Inhibitors via a TR-FRET Assay reconfirm |
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| IC50 | 1315±36 nM |
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| Citation |  PubChem, PC Dose Response confirmation of uHTS for the identification of UBC13 Polyubiquitin Inhibitors via a TR-FRET Assay reconfirm PubChem Bioassay(2011)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| Ubiquitin-conjugating enzyme E2 N |
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| Name: | Ubiquitin-conjugating enzyme E2 N |
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| Synonyms: | BLU | UBE2N | UBE2N_HUMAN | ubiquitin-conjugating enzyme E2 N |
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| Type: | PROTEIN |
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| Mol. Mass.: | 17137.61 |
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| Organism: | Homo sapiens (Human) |
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| Description: | EBI_101440 |
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| Residue: | 152 |
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| Sequence: | MAGLPRRIIKETQRLLAEPVPGIKAEPDESNARYFHVVIAGPQDSPFEGGTFKLELFLPE
EYPMAAPKVRFMTKIYHPNVDKLGRICLDILKDKWSPALQIRTVLLSIQALLSAPNPDDP
LANDVAEQWKTNEAQAIETARAWTRLYAMNNI
|
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|
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| BDBM78543 |
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| n/a |
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| Name | BDBM78543 |
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| Synonyms: | MLS000087827 | N-(2-methyl-4-oxidanylidene-quinazolin-3-yl)-4-propoxy-benzamide | N-(2-methyl-4-oxo-3-quinazolinyl)-4-propoxybenzamide | N-(2-methyl-4-oxoquinazolin-3(4H)-yl)-4-propoxybenzamide | N-(2-methyl-4-oxoquinazolin-3-yl)-4-propoxybenzamide | N-(4-keto-2-methyl-quinazolin-3-yl)-4-propoxy-benzamide | SMR000024047 | cid_3237593 |
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| Type | Small organic molecule |
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| Emp. Form. | C19H19N3O3 |
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| Mol. Mass. | 337.3725 |
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| SMILES | CCCOc1ccc(cc1)C(=O)Nn1c(C)nc2ccccc2c1=O |
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| Structure | 
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