| Reaction Details |
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 | Report a problem with these data |
| Target | Ubiquitin-conjugating enzyme E2 N |
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| Ligand | BDBM78626 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Dose Response confirmation of uHTS for the identification of UBC13 Polyubiquitin Inhibitors via a TR-FRET Assay reconfirm |
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| IC50 | 1246±38 nM |
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| Citation |  PubChem, PC Dose Response confirmation of uHTS for the identification of UBC13 Polyubiquitin Inhibitors via a TR-FRET Assay reconfirm PubChem Bioassay(2011)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| Ubiquitin-conjugating enzyme E2 N |
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| Name: | Ubiquitin-conjugating enzyme E2 N |
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| Synonyms: | BLU | UBE2N | UBE2N_HUMAN | ubiquitin-conjugating enzyme E2 N |
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| Type: | PROTEIN |
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| Mol. Mass.: | 17137.61 |
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| Organism: | Homo sapiens (Human) |
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| Description: | EBI_101440 |
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| Residue: | 152 |
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| Sequence: | MAGLPRRIIKETQRLLAEPVPGIKAEPDESNARYFHVVIAGPQDSPFEGGTFKLELFLPE
EYPMAAPKVRFMTKIYHPNVDKLGRICLDILKDKWSPALQIRTVLLSIQALLSAPNPDDP
LANDVAEQWKTNEAQAIETARAWTRLYAMNNI
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| BDBM78626 |
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| n/a |
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| Name | BDBM78626 |
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| Synonyms: | 2-Amino-4-methyl-thiazole-5-carboxylic acid (1H-indol-3-ylmethylene)-hydrazide | 2-amino-N'-[(Z)-3-indolylidenemethyl]-4-methyl-5-thiazolecarbohydrazide | 2-amino-N'-[(Z)-indol-3-ylidenemethyl]-4-methyl-1,3-thiazole-5-carbohydrazide | 2-amino-N'-[(Z)-indol-3-ylidenemethyl]-4-methyl-thiazole-5-carbohydrazide | 2-azanyl-N'-[(Z)-indol-3-ylidenemethyl]-4-methyl-1,3-thiazole-5-carbohydrazide | MLS000525734 | SMR000116208 | cid_6537515 |
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| Type | Small organic molecule |
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| Emp. Form. | C14H13N5OS |
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| Mol. Mass. | 299.351 |
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| SMILES | Cc1nc(N)sc1C(=O)NN=Cc1c[nH]c2ccccc12 |w:10.10| |
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| Structure | 
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