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TargetDNA dC->dU-editing enzyme APOBEC-3G
LigandBDBM46661
Substrate/Competitorn/a
Meas. Tech.Dose Response confirmation of small molecule APOBEC3G DNA Deaminase Inhibitors via a fluorescence-based single-stranded DNA deaminase assay
Temperature298.15±n/a K
IC50 1950±n/a nM
Commentsextracted
Citation PubChem, PC Dose Response confirmation of small molecule APOBEC3G DNA Deaminase Inhibitors via a fluorescence-based single-stranded DNA deaminase assay PubChem Bioassay(2011)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
DNA dC->dU-editing enzyme APOBEC-3G
Name:DNA dC->dU-editing enzyme APOBEC-3G
Synonyms:ABC3G_HUMAN | APOBEC3G
Type:Enzyme Catalytic Domain
Mol. Mass.:46419.54
Organism:Homo sapiens (Human)
Description:gi_13399304
Residue:384
Sequence:
MKPHFRNTVERMYRDTFSYNFYNRPILSRRNTVWLCYEVKTKGPSRPPLDAKIFRGQVYS
ELKYHPEMRFFHWFSKWRKLHRDQEYEVTWYISWSPCTKCTRDMATFLAEDPKVTLTIFV
ARLYYFWDPDYQEALRSLCQKRDGPRATMKIMNYDEFQHCWSKFVYSQRELFEPWNNLPK
YYILLHIMLGEILRHSMDPPTFTFNFNNEPWVRGRHETYLCYEVERMHNDTWVLLNQRRG
FLCNQAPHKHGFLEGRHAELCFLDVIPFWKLDLDQDYRVTCFTSWSPCFSCAQEMAKFIS
KNKHVSLCIFTARIYDDQGRCQEGLRTLAEAGAKISIMTYSEFKHCWDTFVDHQGCPFQP
WDGLDEHSQDLSGRLRAILQNQEN
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  Blast E-value cutoff:
BDBM46661
n/a
NameBDBM46661
Synonyms:5-(4-methoxyphenyl)-1,2-dihydro-1,2,4-triazole-3-thione | MLS-0013008.0001 | cid_689101
TypeSmall organic molecule
Emp. Form.C9H9N3OS
Mol. Mass.207.252
SMILESCOc1ccc(cc1)-c1n[nH]c(=S)[nH]1
Structure
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