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TargetC-C chemokine receptor type 6
LigandBDBM79992
Substrate/Competitorn/a
Meas. Tech.Dose Response confirmation of small molecule antagonists of the CCR6 receptor: a luminescent beta-arrestin assay
IC50 13900±n/a nM
Citation PubChem, PC Dose Response confirmation of small molecule antagonists of the CCR6 receptor: a luminescent beta-arrestin assay PubChem Bioassay(2011)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
C-C chemokine receptor type 6
Name:C-C chemokine receptor type 6
Synonyms:C-C chemokine receptor type 6 | C-C chemokine receptor type 6 (CCR6) | CCR6 | CCR6_HUMAN | CKRL3 | CMKBR6 | GPR29 | STRL22
Type:Enzyme
Mol. Mass.:42510.84
Organism:Homo sapiens (Human)
Description:P51684
Residue:374
Sequence:
MSGESMNFSDVFDSSEDYFVSVNTSYYSVDSEMLLCSLQEVRQFSRLFVPIAYSLICVFG
LLGNILVVITFAFYKKARSMTDVYLLNMAIADILFVLTLPFWAVSHATGAWVFSNATCKL
LKGIYAINFNCGMLLLTCISMDRYIAIVQATKSFRLRSRTLPRSKIICLVVWGLSVIISS
STFVFNQKYNTQGSDVCEPKYQTVSEPIRWKLLMLGLELLFGFFIPLMFMIFCYTFIVKT
LVQAQNSKRHKAIRVIIAVVLVFLACQIPHNMVLLVTAANLGKMNRSCQSEKLIGYTKTV
TEVLAFLHCCLNPVLYAFIGQKFRNYFLKILKDLWCVRRKYKSSGFSCAGRYSENISRQT
SETADNDNASSFTM
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BDBM79992
n/a
NameBDBM79992
Synonyms:(5-chloranylquinolin-8-yl) 4-methyl-3-nitro-benzoate | (5-chloroquinolin-8-yl) 4-methyl-3-nitrobenzoate | 4-methyl-3-nitro-benzoic acid (5-chloro-8-quinolyl) ester | 4-methyl-3-nitrobenzoic acid (5-chloro-8-quinolinyl) ester | 5-chloro-8-quinolinyl 4-methyl-3-nitrobenzoate | MLS000576307 | SMR000197947 | cid_887191
TypeSmall organic molecule
Emp. Form.C17H11ClN2O4
Mol. Mass.342.733
SMILESCc1ccc(cc1[N+]([O-])=O)C(=O)Oc1ccc(Cl)c2cccnc12
Structure
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