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TargetC-C chemokine receptor type 6
LigandBDBM80075
Substrate/Competitorn/a
Meas. Tech.Dose Response confirmation of small molecule antagonists of the CCR6 receptor: a luminescent beta-arrestin assay
IC50>66600±n/a nM
Citation PubChem, PC Dose Response confirmation of small molecule antagonists of the CCR6 receptor: a luminescent beta-arrestin assay PubChem Bioassay(2011)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
C-C chemokine receptor type 6
Name:C-C chemokine receptor type 6
Synonyms:C-C chemokine receptor type 6 | C-C chemokine receptor type 6 (CCR6) | CCR6 | CCR6_HUMAN | CKRL3 | CMKBR6 | GPR29 | STRL22
Type:Enzyme
Mol. Mass.:42510.84
Organism:Homo sapiens (Human)
Description:P51684
Residue:374
Sequence:
MSGESMNFSDVFDSSEDYFVSVNTSYYSVDSEMLLCSLQEVRQFSRLFVPIAYSLICVFG
LLGNILVVITFAFYKKARSMTDVYLLNMAIADILFVLTLPFWAVSHATGAWVFSNATCKL
LKGIYAINFNCGMLLLTCISMDRYIAIVQATKSFRLRSRTLPRSKIICLVVWGLSVIISS
STFVFNQKYNTQGSDVCEPKYQTVSEPIRWKLLMLGLELLFGFFIPLMFMIFCYTFIVKT
LVQAQNSKRHKAIRVIIAVVLVFLACQIPHNMVLLVTAANLGKMNRSCQSEKLIGYTKTV
TEVLAFLHCCLNPVLYAFIGQKFRNYFLKILKDLWCVRRKYKSSGFSCAGRYSENISRQT
SETADNDNASSFTM
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM80075
n/a
NameBDBM80075
Synonyms:7-bromanyl-6-methoxy-quinoline-5,8-dione | 7-bromo-6-methoxy-quinoline-5,8-quinone | 7-bromo-6-methoxyquinoline-5,8-dione | MLS002703741 | SMR001570458 | cid_265935
TypeSmall organic molecule
Emp. Form.C10H6BrNO3
Mol. Mass.268.064
SMILESCOC1=C(Br)C(=O)c2ncccc2C1=O |c:2|
Structure
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