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| Reaction Details | |||
|---|---|---|---|
 | Report a problem with these data | ||
| Target | cAMP-dependent protein kinase type II-beta regulatory subunit | ||
| Ligand | BDBM81291 | ||
| Substrate/Competitor | n/a | ||
| Meas. Tech. | Fluorescence polarization-based biochemical high throughput dose response assay for activators of the Protein Kinase A-R2B (PKA-R2B) complex | ||
| EC50 | 50.49±n/a nM | ||
| Citation |  PubChem, PC Fluorescence polarization-based biochemical high throughput dose response assay for activators of the Protein Kinase A-R2B (PKA-R2B) complex PubChem Bioassay(2011)[AID] | ||
| More Info.: | Get all data from this article, Solution Info, Assay Method | ||
| cAMP-dependent protein kinase type II-beta regulatory subunit | |||
| Name: | cAMP-dependent protein kinase type II-beta regulatory subunit | ||
| Synonyms: | KAP3_HUMAN | PRKAR2B | ||
| Type: | PROTEIN | ||
| Mol. Mass.: | 46282.41 | ||
| Organism: | Homo sapiens (Human) | ||
| Description: | EBI_11972 | ||
| Residue: | 418 | ||
| Sequence: |
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| BDBM81291 | |||
| n/a | |||
| Name | BDBM81291 | ||
| Synonyms: | 8-(4-Chlorophenylthio)adenosine 3',5'-cyclic monophosphate sodium salt | MLS002153200 | SMR000326853 | cid_23672705 | sodium;(4aR,6R,7R,7aS)-6-[6-amino-8-(4-chlorophenyl)sulfanylpurin-9-yl]-2-oxido-2-oxo-4a,6,7,7a-tetrahydro-4H-furo[3,2-d][1,3,2]dioxaphosphinin-7-ol | sodium;(4aR,6R,7R,7aS)-6-[6-amino-8-[(4-chlorophenyl)thio]-9-purinyl]-2-oxido-2-oxo-4a,6,7,7a-tetrahydro-4H-furo[3,2-d][1,3,2]dioxaphosphorin-7-ol | sodium;(4aR,6R,7R,7aS)-6-[6-amino-8-[(4-chlorophenyl)thio]purin-9-yl]-2-keto-2-oxido-4a,6,7,7a-tetrahydro-4H-furo[3,2-d][1,3,2]dioxaphosphorin-7-ol | sodium;(4aR,6R,7R,7aS)-6-[6-azanyl-8-(4-chlorophenyl)sulfanyl-purin-9-yl]-2-oxidanidyl-2-oxidanylidene-4a,6,7,7a-tetrahydro-4H-furo[3,2-d][1,3,2]dioxaphosphinin-7-ol | ||
| Type | Small organic molecule | ||
| Emp. Form. | C16H14ClN5O6PS | ||
| Mol. Mass. | 470.805 | ||
| SMILES | Nc1ncnc2n([C@@H]3O[C@@H]4COP([O-])(=O)O[C@H]4[C@H]3O)c(Sc3ccc(Cl)cc3)nc12 | ||
| Structure | 
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