Reaction Details | |||
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Target | cAMP-dependent protein kinase type II-beta regulatory subunit | ||
Ligand | BDBM81290 | ||
Substrate/Competitor | n/a | ||
Meas. Tech. | Counterscreen for activators of the Protein Kinase A-R1A (PKA-R1A) complex | ||
EC50 | 11726±n/a nM | ||
Citation | PubChem, PC Counterscreen for activators of the Protein Kinase A-R1A (PKA-R1A) complex: fluorescence polarization-based biochemical high throughput dose response assay to identify activators of the Protein Kinase A-R2B (PKA-R2B) complex PubChem Bioassay(2011)[AID] | ||
More Info.: | Get all data from this article, Solution Info, Assay Method | ||
cAMP-dependent protein kinase type II-beta regulatory subunit | |||
Name: | cAMP-dependent protein kinase type II-beta regulatory subunit | ||
Synonyms: | KAP3_HUMAN | PRKAR2B | ||
Type: | PROTEIN | ||
Mol. Mass.: | 46282.41 | ||
Organism: | Homo sapiens (Human) | ||
Description: | EBI_11972 | ||
Residue: | 418 | ||
Sequence: |
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BDBM81290 | |||
n/a | |||
Name | BDBM81290 | ||
Synonyms: | MLS001148197 | N6,2'-O-DIBUTYRYLADENOSINE-3',5'-CYCLIC MONOPHOSPHATE SODIUM SALT | SMR000058940 | cid_23663967 | sodium;[(4aR,6R,7R,7aR)-6-[6-(butanoylamino)purin-9-yl]-2-oxidanidyl-2-oxidanylidene-4a,6,7,7a-tetrahydro-4H-furo[3,2-d][1,3,2]dioxaphosphinin-7-yl] butanoate | sodium;[(4aR,6R,7R,7aR)-6-[6-(butanoylamino)purin-9-yl]-2-oxido-2-oxo-4a,6,7,7a-tetrahydro-4H-furo[3,2-d][1,3,2]dioxaphosphinin-7-yl] butanoate | sodium;butanoic acid [(4aR,6R,7R,7aR)-2-oxido-2-oxo-6-[6-(1-oxobutylamino)-9-purinyl]-4a,6,7,7a-tetrahydro-4H-furo[3,2-d][1,3,2]dioxaphosphorin-7-yl] ester | sodium;butyric acid [(4aR,6R,7R,7aR)-6-(6-butyramidopurin-9-yl)-2-keto-2-oxido-4a,6,7,7a-tetrahydro-4H-furo[3,2-d][1,3,2]dioxaphosphorin-7-yl] ester | sodium;butyric acid [(4aR,6R,7R,7aR)-6-(6-butyramidopurin-9-yl)-2-keto-2-oxido-4a,6,7,7a-tetrahydro-4H-furo[3,2-d][1,3,2]dioxaphosphorin-7-yl] ester;hydrate | ||
Type | Small organic molecule | ||
Emp. Form. | C18H23N5O8P | ||
Mol. Mass. | 468.3782 | ||
SMILES | CCCC(=O)Nc1ncnc2n(cnc12)[C@@H]1O[C@@H]2COP([O-])(=O)O[C@H]2[C@H]1OC(=O)CCC | ||
Structure |