| Reaction Details |
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 | Report a problem with these data |
| Target | Leukotriene B4 receptor 2 |
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| Ligand | BDBM81522 |
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| Substrate/Competitor | n/a |
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| Ki | 24±n/a nM |
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| Comments | PDSP_496 |
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| Citation |  Jackson, RH; Morrissey, MM; Sills, MA; Jarvis, MF Comparison of antagonist and agonist binding to the leukotriene B4 receptor intact human polymorphonuclear neutrophils (PMN). J Pharmacol Exp Ther262:80-9 (1992) [PubMed] |
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| More Info.: | Get all data from this article |
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| Leukotriene B4 receptor 2 |
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| Name: | Leukotriene B4 receptor 2 |
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| Synonyms: | BLT2R | BLTR2 | LT4R2_HUMAN | LTB4 receptor JULF2 | LTB4-R 2 | LTB4-R2 | LTB4R2 | LTB4R2 protein | Leukotriene B4 | Leukotriene B4 R2 | Leukotriene B4 receptor | Leukotriene B4 receptor 2 | Leukotriene B4 receptor BLT2 | Leukotriene b1 | Seven transmembrane receptor BLTR2 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 37964.86 |
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| Organism: | Homo sapiens (Human) |
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| Description: | Leukotriene 2 0 HUMAN::Q9NPC1 |
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| Residue: | 358 |
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| Sequence: | MSVCYRPPGNETLLSWKTSRATGTAFLLLAALLGLPGNGFVVWSLAGWRPARGRPLAATL
VLHLALADGAVLLLTPLFVAFLTRQAWPLGQAGCKAVYYVCALSMYASVLLTGLLSLQRC
LAVTRPFLAPRLRSPALARRLLLAVWLAALLLAVPAAVYRHLWRDRVCQLCHPSPVHAAA
HLSLETLTAFVLPFGLMLGCYSVTLARLRGARWGSGRHGARVGRLVSAIVLAFGLLWAPY
HAVNLLQAVAALAPPEGALAKLGGAGQAARAGTTALAFFSSSVNPVLYVFTAGDLLPRAG
PRFLTRLFEGSGEARGGGRSREGTMELRTTPQLKVVGQGRGNGDPGGGMEKDGPEWDL
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| BDBM81522 |
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| n/a |
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| Name | BDBM81522 |
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| Synonyms: | CGS 23130 |
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| Type | Small organic molecule |
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| Emp. Form. | C29H30O7 |
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| Mol. Mass. | 490.5443 |
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| SMILES | COc1ccc(\C=C\CCCCOc2ccc(Oc3cccc(c3)C(O)=O)cc2CCC(O)=O)cc1 |
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| Structure | 
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