| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Somatostatin receptor type 4 |
|---|
| Ligand | BDBM50059090 |
|---|
| Substrate/Competitor | n/a |
|---|
| Ki | 0.18±n/a nM |
|---|
| Comments | PDSP_1734 |
|---|
| Citation |  O'Carroll, AM; Lolait, SJ; König, M; Mahan, LC Molecular cloning and expression of a pituitary somatostatin receptor with preferential affinity for somatostatin-28. Mol Pharmacol42:939-46 (1992) [PubMed] |
|---|
| More Info.: | Get all data from this article |
|---|
| |
| Somatostatin receptor type 4 |
|---|
| Name: | Somatostatin receptor type 4 |
|---|
| Synonyms: | SOMATOSTATIN SST4 | SSR4_RAT | Somatostatin receptor | Somatostatin receptor type 4 | Sstr4 |
|---|
| Type: | Enzyme Catalytic Domain |
|---|
| Mol. Mass.: | 42096.84 |
|---|
| Organism: | RAT |
|---|
| Description: | SOMATOSTATIN SST4 SSTR4 RAT::P30937 |
|---|
| Residue: | 384 |
|---|
| Sequence: | MNTPATLPLGGEDTTWTPGINASWAPDEEEDAVRSDGTGTAGMVTIQCIYALVCLVGLVG
NALVIFVILRYAKMKTATNIYLLNLAVADELFMLSVPFVASAAALRHWPFGAVLCRAVLS
VDGLNMFTSVFCLTVLSVDRYVAVVHPLRAATYRRPSVAKLINLGVWLASLLVTLPIAVF
ADTRPARGGEAVACNLHWPHPAWSAVFVIYTFLLGFLLPVLAIGLCYLLIVGKMRAVALR
AGWQQRRRSEKKITRLVLMVVTVFVLCWMPFYVVQLLNLFVTSLDATVNHVSLILSYANS
CANPILYGFLSDNFRRSFQRVLCLRCCLLETTGGAEEEPLDYYATALKSRGGPGCICPPL
PCQQEPMQAEPACKRVPFTKTTTF
|
|
|
|---|
| BDBM50059090 |
|---|
| n/a |
|---|
| Name | BDBM50059090 |
|---|
| Synonyms: | 10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionylamino)-16-benzyl-7-(1-hydroxy-ethyl)-13-(1H-indol-3-ylmethyl)-6,9,12,15,18-pentaoxo-1,2-dithia-5,8,11,14,17-pentaaza-cycloicosane-4-carboxylic acid (2-hydroxy-1-hydroxymethyl-propyl)-amide | CHEMBL405598 | SMS 201-995 | octreotide |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C49H66N10O10S2 |
|---|
| Mol. Mass. | 1019.239 |
|---|
| SMILES | CC(O)[C@H](CO)NC(=O)[C@@H]1CSSCC(NC(=O)C(N)Cc2ccccc2)C(=O)N[C@H](Cc2ccccc2)C(=O)N[C@H](Cc2c[nH]c3ccccc23)C(=O)N[C@H](CCCCN)C(=O)N[C@H](C(C)O)C(=O)N1 |
|---|
| Structure | 
|
|---|
Search and Browse
