| Reaction Details |
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 | Report a problem with these data |
| Target | Gastrin/cholecystokinin type B receptor |
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| Ligand | BDBM81869 |
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| Substrate/Competitor | n/a |
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| Ki | 510±n/a nM |
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| Comments | PDSP_2194 |
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| Citation |  Lin, CW; Shiosaki, K; Miller, TR; Witte, DG; Bianchi, BR; Wolfram, CA; Kopecka, H; Craig, R; Wagenaar, F; Nadzan, AM Characterization of two novel cholecystokinin tetrapeptide (30-33) analogues, A-71623 and A-70874, that exhibit high potency and selectivity for cholecystokinin-A receptors. Mol Pharmacol39:346-51 (1991) [PubMed] |
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| More Info.: | Get all data from this article |
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| Gastrin/cholecystokinin type B receptor |
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| Name: | Gastrin/cholecystokinin type B receptor |
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| Synonyms: | CCKBR | Cholecystokinin A |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 48683.10 |
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| Organism: | GUINEA PIG |
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| Description: | Cholecystokinin A CCKBR GUINEA PIG::H0VZC5 |
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| Residue: | 450 |
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| Sequence: | MELLKLNRSLQGPGPGPGAPLCRPAGPLLNSSGAGNVSCETPRIRGAGTRVKSMAILFNV
TSLLSCWNKYRIIKVLGLSRRLRTVTKAFLLSLAVSDLLLAVACMPFTLLPNLMGTFIFG
TVICKAVSYLMGVSVSVSTLSLVAIALERYSAICRPLQARVWQTRSHAARVILATWLLSG
LLMVPYPVYTAVQPVGPRVLQCVHRWPNARVRQTWSVLLLLLLFFVPGVVMAVAYGLISR
ELYLGLRFDGDADSESQSRVRGPGGLSGSAPGPAHQNGRCRPESGLSGEDSDGCYVQLPR
SRPALELSALAASTPAPGPGPRPTQAKLLAKKRVVRMLLVIVVLFFLCWLPVYSANTWRA
FDGPGAHRALSGAPISFIHLLSYASACVNPLVYCFMHRRFRQACLDTCARCCPRPPRARP
RPLPEEDPPTPSIASLSRLSYTTISTLGPG
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| BDBM81869 |
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| n/a |
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| Name | BDBM81869 |
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| Synonyms: | A-57282 |
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| Type | n/a |
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| Emp. Form. | C43H53N7O10 |
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| Mol. Mass. | 827.9218 |
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| SMILES | CC(C)(C)OC(=O)NC(Cc1c[nH]c2ccccc12)C(=O)N(C(=O)C(N)Cc1ccccc1)C(=O)C(CC(O)=O)NC(=O)C(N)CCCCNC(=O)OCc1ccccc1 |
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| Structure | 
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