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TargetP2Y purinoceptor 2
LigandBDBM10847
Substrate/Competitorn/a
Ki 4550±n/a nM
CommentsPDSP_2649
Citation Klotz, KNVogt, HTawfik-Schlieper, H Comparison of A1 adenosine receptors in brain from different species by radioligand binding and photoaffinity labelling. Naunyn Schmiedebergs Arch Pharmacol343:196-201 (1991) [PubMed]  Article
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P2Y purinoceptor 2
Name:P2Y purinoceptor 2
Synonyms:ADENOSINE A1 | ADENOSINE A1 high | ADENOSINE A1 low | ADORA1 | P2RY2 | P2RY2_CRIGR | P2Y purinoceptor 2
Type:Enzyme Catalytic Domain
Mol. Mass.:18813.49
Organism:HAMSTER
Description:ADENOSINE A1 ADORA1 HAMSTER::P58825
Residue:166
Sequence:
VHRCLGVLRPLHSLRWGRARYARRVAAVVWVLVLACQAPVLYFVTTSVRGTRITCHDTSA
RELFSHFVAYSSVMLSLLFAVPFSVILVCYVLMARRLLKPAYGTTGGLPRAKRKSVRTIA
LVLAVFTLCFLPFHVTRTLYYSFRSLDLSCHTLNAINMAYKITRPL
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  Blast E-value cutoff:
BDBM10847
n/a
NameBDBM10847
Synonyms:1,3-dimethyl-2,3,6,7-tetrahydro-1H-purine-2,6-dione | 1,3-dimethyl-7H-purine-2,6-dione | Afonilum | Aminophyllin | Aminophylline | CHEMBL190 | Cardophyllin | Euphylline | Theophy-lline | Theophylline | Theophylline (1,3-dimethylxanthine)
TypeSmall organic molecule
Emp. Form.C7H8N4O2
Mol. Mass.180.164
SMILESCn1c2nc[nH]c2c(=O)n(C)c1=O
Structure
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