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TargetP2Y purinoceptor 2
LigandBDBM50008415
Substrate/Competitorn/a
Ki 0.39±n/a nM
CommentsPDSP_2055
Citation Klotz, KNVogt, HTawfik-Schlieper, H Comparison of A1 adenosine receptors in brain from different species by radioligand binding and photoaffinity labelling. Naunyn Schmiedebergs Arch Pharmacol343:196-201 (1991) [PubMed]  Article
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P2Y purinoceptor 2
Name:P2Y purinoceptor 2
Synonyms:ADENOSINE A1 | ADENOSINE A1 high | ADENOSINE A1 low | ADORA1 | P2RY2 | P2RY2_CRIGR | P2Y purinoceptor 2
Type:Enzyme Catalytic Domain
Mol. Mass.:18813.49
Organism:HAMSTER
Description:ADENOSINE A1 ADORA1 HAMSTER::P58825
Residue:166
Sequence:
VHRCLGVLRPLHSLRWGRARYARRVAAVVWVLVLACQAPVLYFVTTSVRGTRITCHDTSA
RELFSHFVAYSSVMLSLLFAVPFSVILVCYVLMARRLLKPAYGTTGGLPRAKRKSVRTIA
LVLAVFTLCFLPFHVTRTLYYSFRSLDLSCHTLNAINMAYKITRPL
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BDBM50008415
n/a
NameBDBM50008415
Synonyms:2-(2-Chloro-6-cyclopentylamino-purin-9-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol | 2-[2-chloro-6-(cyclopentylamino)-9H-purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol | CCPA
TypeSmall organic molecule
Emp. Form.C15H20ClN5O4
Mol. Mass.369.803
SMILESOCC1OC(C(O)C1O)n1cnc2c(NC3CCCC3)nc(Cl)nc12
Structure
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