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Targetkappa-type opioid receptor isoform 1
LigandBDBM81935
Substrate/Competitorn/a
Ki 0.4±n/a nM
CommentsPDSP_1351
Citation Benyhe, SVarga, EHepp, JMagyar, ABorsodi, AWollemann, M Characterization of kappa 1 and kappa 2 opioid binding sites in frog (Rana esculenta) brain membrane preparation. Neurochem Res15:899-904 (1990) [PubMed]  Article
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kappa-type opioid receptor isoform 1
Name:kappa-type opioid receptor isoform 1
Synonyms:OPIATE Kappa | OPRK1
Type:Enzyme Catalytic Domain
Mol. Mass.:42362.28
Organism:Frog
Description:F7A0F2
Residue:375
Sequence:
MCFNLTMKKKKECCAPACPSSCFPNTSWLLGWDDHDNVSAYPDLPLNEGNHTSISPTISV
IITAVYSMVFVVGLVGNALVMFVIIRYTKMKTATNIYIFNLALADALVTTTMPFQSTSFL
MNSWPFGDVLCKIVVSIDYYNMFTSIFTLTMMSVDRYIAVCHPVKALDFRTPLKAKCINI
CIWMLSSSVGISAIVLGGTKISDGSTECALQFPTHYWYWDTVMKMCVFIFAFIIPVFIIT
ICYTLMILRLKSVRLLSGSREKDRNLRRITRLVLVVVAVFIVCWTPIHIFVLVEALVDVP
QSIAVVSIYYFCIALGYTNSSLNPILYAFLDENFKRCFKDFCFPSKHRLDRQPNSRVGNT
VQDPACNRHGSQKPV
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM81935
n/a
NameBDBM81935
Synonyms:CAS_105618-26-6 | NSC_3034416 | Nor-BNI
TypeSmall organic molecule
Emp. Form.C40H43N3O6
Mol. Mass.661.7859
SMILESOc1ccc2CC(C3CC3)N3CCC45C(Oc1c24)c1[nH]c2C4Oc6c7c(CC(C8CC8)N8CCC47C(O)(C8)Cc2c1CC5(O)C3)ccc6O |TLB:7:6:12.11:44.42,43:42:6.5.4.17:12.11,28:27:35.37:32.33,THB:23:24:35.37:32.33,45:25:35.37:32.33,41:42:6.5.4.17:12.11,16:17:12.11:44.42,3:4:12.11:44.42,36:35:32.33:25.24.26.27|
Structure
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