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Reaction Details
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TargetNorepinephrine transporter
LigandBDBM50021217
Substrate/Competitorn/a
Ki 0.79±n/a nM
CommentsPDSP_3888
Citation Hyttel, JLarsen, JJ Neurochemical profile of Lu 19-005, a potent inhibitor of uptake of dopamine, noradrenaline, and serotonin. J Neurochem44:1615-22 (1985) [PubMed]  Article
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Norepinephrine transporter
Name:Norepinephrine transporter
Synonyms:n/a
Type:Enzyme Catalytic Domain
Mol. Mass.:2082.45
Organism:RAT
Description:Norepinephrine transporter 0 RAT::Q9JIA2
Residue:19
Sequence:
MLLARMKPQVQPELGGADQ
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BDBM50021217
n/a
NameBDBM50021217
Synonyms:CHEMBL52247 | Talsupram | [3-(3,3-Dimethyl-1-phenyl-1,3-dihydro-benzo[c]thiophen-1-yl)-propyl]-methyl-amine(Talsupram)
TypeSmall organic molecule
Emp. Form.C20H25NS
Mol. Mass.311.484
SMILESCNCCCC1(SC(C)(C)c2ccccc12)c1ccccc1
Structure
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