| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Adenosine receptor A1 |
|---|
| Ligand | BDBM50004464 |
|---|
| Substrate/Competitor | n/a |
|---|
| Ki | 910±n/a nM |
|---|
| Comments | PDSP_2892 |
|---|
| Citation |  Hutchison, AJ; Webb, RL; Oei, HH; Ghai, GR; Zimmerman, MB; Williams, M CGS 21680C, an A2 selective adenosine receptor agonist with preferential hypotensive activity. J Pharmacol Exp Ther251:47-55 (1989) [PubMed] |
|---|
| More Info.: | Get all data from this article |
|---|
| |
| Adenosine receptor A1 |
|---|
| Name: | Adenosine receptor A1 |
|---|
| Synonyms: | AA1R_RAT | ADENOSINE A1 | ADENOSINE A1 high | ADENOSINE A1 low | Adenosine A1 receptor (A1) | Adenosine receptor | Adenosine receptors A1 | Adora1 |
|---|
| Type: | Protein |
|---|
| Mol. Mass.: | 36704.13 |
|---|
| Organism: | Rattus norvegicus (rat) |
|---|
| Description: | n/a |
|---|
| Residue: | 326 |
|---|
| Sequence: | MPPYISAFQAAYIGIEVLIALVSVPGNVLVIWAVKVNQALRDATFCFIVSLAVADVAVGA
LVIPLAILINIGPQTYFHTCLMVACPVLILTQSSILALLAIAVDRYLRVKIPLRYKTVVT
QRRAAVAIAGCWILSLVVGLTPMFGWNNLSVVEQDWRANGSVGEPVIKCEFEKVISMEYM
VYFNFFVWVLPPLLLMVLIYLEVFYLIRKQLNKKVSASSGDPQKYYGKELKIAKSLALIL
FLFALSWLPLHILNCITLFCPTCQKPSILIYIAIFLTHGNSAMNPIVYAFRIHKFRVTFL
KIWNDHFRCQPKPPIDEDLPEEKAED
|
|
|
|---|
| BDBM50004464 |
|---|
| n/a |
|---|
| Name | BDBM50004464 |
|---|
| Synonyms: | (CV 1808) 2-(6-Amino-2-phenylamino-purin-9-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol | 2-(6-Amino-2-phenylamino-purin-9-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol | CV 1808 | CV-1808 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C16H18N6O4 |
|---|
| Mol. Mass. | 358.3519 |
|---|
| SMILES | Nc1nc(Nc2ccccc2)nc2n(cnc12)[C@@H]1O[C@H](CO)[C@H](O)C1O |
|---|
| Structure | 
|
|---|
Search and Browse
