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TargetAlpha-1A adrenergic receptor
LigandBDBM84342
Substrate/Competitorn/a
Ki 30±n/a nM
CommentsPDSP_238
Citation Jones, SBSmith, JMJones, AWBylund, DB Alpha-1 adrenergic receptor binding in aortas from rat and dog: comparison of [3H]prazosin and beta-iodo-[125I]-4-hydroxyphenyl-ethyl-aminomethyl-tetralone. J Pharmacol Exp Ther241:875-81 (1987) [PubMed]
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Alpha-1A adrenergic receptor
Name:Alpha-1A adrenergic receptor
Synonyms:ADA1A_CANLF | ADRA1A | ADRA1C | adrenergic Alpha1
Type:Enzyme Catalytic Domain
Mol. Mass.:32268.65
Organism:Dog
Description:adrenergic Alpha1 0 Dog::O77621
Residue:295
Sequence:
MVFLSGNASDSSNCTHPPAPVNISKAILLGVILGGLIIFGVLGNILVILSVACHRHLHSV
THYYIVNLAVADLLLTSTVLPFSAIFEILGYWAFGRVFCNIWAAVDVLCCTASIMGLCII
SIDRYIGVSYPLRYPTIVTQKRGLMALLCVWALSLVISIGPLFGWRQPAPEDETICQITE
EPGYVLFSALGSFYVPLTIILVMYCRVYVVAKRESRGLKSGLKTDKSDSEQVTLRIHRKN
APVGGTGVSSAKNKTHFSVRLLKFSREKKAAKTLGIVVGCFVLCWLPFFLVMPIG
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BDBM84342
n/a
NameBDBM84342
Synonyms:4-[1-hydroxy-2-(methylamino)ethyl]benzene-1,2-diol | 4-[1-hydroxy-2-(methylamino)ethyl]benzene-1,2-diol, 1 | 4-[1-hydroxy-2-(methylamino)ethyl]benzene-1,2-diol;hydrochloride | 4-[1-hydroxy-2-(methylamino)ethyl]pyrocatechol;hydrochloride | 4-[2-(methylamino)-1-oxidanyl-ethyl]benzene-1,2-diol;hydrochloride | DL-ADRENALINE HYDROCHLORIDE | EPINEPHRINE | EPINEPHRINE,(+) | MLS001333244 | SMR000058236 | cid_5924
TypeSmall organic molecule
Emp. Form.C9H13NO3
Mol. Mass.183.2044
SMILESCNCC(O)c1ccc(O)c(O)c1
Structure
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