| Reaction Details |
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 | Report a problem with these data |
| Target | Thromboxane A2 receptor |
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| Ligand | BDBM50002765 |
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| Substrate/Competitor | n/a |
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| Ki | 1404±n/a nM |
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| Comments | PDSP_401 |
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| Citation |  Hedberg, A; Hall, SE; Ogletree, ML; Harris, DN; Liu, EC Characterization of [5,6-3H]SQ 29,548 as a high affinity radioligand, binding to thromboxane A2/prostaglandin H2-receptors in human platelets. J Pharmacol Exp Ther245:786-92 (1988) [PubMed] |
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| More Info.: | Get all data from this article |
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| Thromboxane A2 receptor |
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| Name: | Thromboxane A2 receptor |
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| Synonyms: | Prostanoid TP receptor | TA2R_HUMAN | TBXA2R | TXA2-R | Thromboxane | Thromboxane A2 receptor | Thromboxane Beta |
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| Type: | Enyzme |
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| Mol. Mass.: | 37445.28 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P21731 |
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| Residue: | 343 |
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| Sequence: | MWPNGSSLGPCFRPTNITLEERRLIASPWFAASFCVVGLASNLLALSVLAGARQGGSHTR
SSFLTFLCGLVLTDFLGLLVTGTIVVSQHAALFEWHAVDPGCRLCRFMGVVMIFFGLSPL
LLGAAMASERYLGITRPFSRPAVASQRRAWATVGLVWAAALALGLLPLLGVGRYTVQYPG
SWCFLTLGAESGDVAFGLLFSMLGGLSVGLSFLLNTVSVATLCHVYHGQEAAQQRPRDSE
VEMMAQLLGIMVVASVCWLPLLVFIAQTVLRNPPAMSPAGQLSRTTEKELLIYLRVATWN
QILDPWVYILFRRAVLRRLQPRLSTRPRSLSLQPQLTQRSGLQ
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| BDBM50002765 |
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| n/a |
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| Name | BDBM50002765 |
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| Synonyms: | BM 13177 | BM-13177 | CHEMBL8273 | Sulotroban | [4-(2-Benzenesulfonylamino-ethyl)-phenoxy]-acetic acid | [4-(2-Benzenesulfonylamino-ethyl)-phenoxy]-acetic acid (BM 13177) | [4-(2-Benzenesulfonylamino-ethyl)-phenoxy]-acetic acid(sulotroban) |
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| Type | Small organic molecule |
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| Emp. Form. | C16H17NO5S |
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| Mol. Mass. | 335.375 |
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| SMILES | OC(=O)COc1ccc(CCNS(=O)(=O)c2ccccc2)cc1 |
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| Structure | 
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