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TargetSigma non-opioid intracellular receptor 1
LigandBDBM50001031
Substrate/Competitorn/a
Ki 229±n/a nM
CommentsPDSP_1714
Citation Mendelsohn, LGKalra, VJohnson, BGKerchner, GA Sigma opioid receptor: characterization and co-identity with the phencyclidine receptor. J Pharmacol Exp Ther233:597-602 (1985) [PubMed]
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Sigma non-opioid intracellular receptor 1
Name:Sigma non-opioid intracellular receptor 1
Synonyms:Opioid receptor | Oprs1 | SGMR1_RAT | Sigma | Sigma non-opioid intracellular receptor 1 | Sigma opioid receptor | Sigma-1 | Sigmar1
Type:Enzyme Catalytic Domain
Mol. Mass.:25266.54
Organism:RAT
Description:Q9R0C9
Residue:223
Sequence:
MPWAVGRRWAWITLFLTIVAVLIQAVWLWLGTQSFVFQREEIAQLARQYAGLDHELAFSR
LIVELRRLHPGHVLPDEELQWVFVNAGGWMGAMCLLHASLSEYVLLFGTALGSHGHSGRY
WAEISDTIISGTFHQWREGTTKSEVYYPGETVVHGPGEATAVEWGPNTWMVEYGRGVIPS
TLAFALSDTIFSTQDFLTLFYTLRAYARGLRLELTTYLFGQDP
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BDBM50001031
n/a
NameBDBM50001031
Synonyms:3-Allyl-6,11-dimethyl-1,2,3,4,5,6-hexahydro-2,6-methano-benzo[d]azocin-8-ol | CHEMBL330376 | SKF 10,047 (+) | SKF 10,047 (-) | SKF 10047
TypeSmall organic molecule
Emp. Form.C17H23NO
Mol. Mass.257.3706
SMILESC[C@H]1[C@H]2Cc3ccc(O)cc3[C@@]1(C)CCN2CC=C |TLB:16:15:1:10.4.3|
Structure
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