| Reaction Details |
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 | Report a problem with these data |
| Target | Norepinephrine transporter |
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| Ligand | BDBM22417 |
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| Substrate/Competitor | n/a |
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| Ki | 3.4±n/a nM |
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| Comments | PDSP_1153 |
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| Citation |  Wong, DT; Threlkeld, PG; Best, KL; Bymaster, FP A new inhibitor of norepinephrine uptake devoid of affinity for receptors in rat brain. J Pharmacol Exp Ther222:61-5 (1982) [PubMed] |
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| More Info.: | Get all data from this article |
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| Norepinephrine transporter |
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| Name: | Norepinephrine transporter |
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| Synonyms: | n/a |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 2082.45 |
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| Organism: | RAT |
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| Description: | Norepinephrine transporter 0 RAT::Q9JIA2 |
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| Residue: | 19 |
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| Sequence: | |
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| BDBM22417 |
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| n/a |
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| Name | BDBM22417 |
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| Synonyms: | 3-(2-methoxyphenoxy)-N-methyl-3-phenylpropan-1-amine | CHEMBL295467 | LY 135252 | LY 94939 | LY135252 | LY139602 | Nisoxetine | Nisoxetine Inhibitor | US9944618, Compound ID No. 177 | [3-(2-methoxyphenoxy)-3-phenylpropyl](methyl)amine | [3H]Nisoxetine |
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| Type | radiolabeled ligand |
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| Emp. Form. | C17H21NO2 |
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| Mol. Mass. | 271.3541 |
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| SMILES | CNCCC(Oc1ccccc1OC)c1ccccc1 |
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| Structure | 
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