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TargetNorepinephrine transporter
LigandBDBM22417
Substrate/Competitorn/a
Ki 1±n/a nM
CommentsPDSP_1330
Citation Wong DTThrelkeld PGBest KLBymaster FP A new inhibitor of norepinephrine uptake devoid of affinity for receptors in rat brain. J Pharmacol Exp Ther 222:61-5 (1982) [PubMed]
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Norepinephrine transporter
Name:Norepinephrine transporter
Synonyms:n/a
Type:Enzyme Catalytic Domain
Mol. Mass.:2082.45
Organism:RAT
Description:Norepinephrine transporter 0 RAT::Q9JIA2
Residue:19
Sequence:
MLLARMKPQVQPELGGADQ
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  Blast E-value cutoff:
BDBM22417
n/a
NameBDBM22417
Synonyms:3-(2-methoxyphenoxy)-N-methyl-3-phenylpropan-1-amine | CHEMBL295467 | LY 135252 | LY 94939 | LY135252 | LY139602 | Nisoxetine | Nisoxetine Inhibitor | [3-(2-methoxyphenoxy)-3-phenylpropyl](methyl)amine | [3H]NISOXETINE | [3H]Nisoxetine | nisoxetine
Typeradiolabeled ligand
Emp. Form.C17H21NO2
Mol. Mass.271.3541
SMILESCNCCC(Oc1ccccc1OC)c1ccccc1
Structure
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