| Reaction Details |
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 | Report a problem with these data |
| Target | Prostacyclin receptor |
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| Ligand | BDBM82098 |
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| Substrate/Competitor | n/a |
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| Ki | 735±n/a nM |
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| Comments | PDSP_5305 |
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| Citation |  Blair, IA; MacDermot, J The binding of [3H]-prostacyclin to membranes of a neuronal somatic hybrid. Br J Pharmacol72:435-41 (1981) [PubMed] Article |
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| More Info.: | Get all data from this article |
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| Prostacyclin receptor |
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| Name: | Prostacyclin receptor |
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| Synonyms: | PGI receptor | PI2R_HUMAN | PRIPR | PTGIR | Prostacyclin (IP) Receptor | Prostacyclin receptor | Prostaglandin I | Prostaglandin I2 | Prostaglandin I2 receptor | Prostanoid IP receptor |
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| Type: | G Protein-Coupled Receptor (GPCR) |
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| Mol. Mass.: | 40968.22 |
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| Organism: | Homo sapiens (Human) |
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| Description: | The membranes prepared from human platelet were used in binding assay. |
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| Residue: | 386 |
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| Sequence: | MADSCRNLTYVRGSVGPATSTLMFVAGVVGNGLALGILSARRPARPSAFAVLVTGLAATD
LLGTSFLSPAVFVAYARNSSLLGLARGGPALCDAFAFAMTFFGLASMLILFAMAVERCLA
LSHPYLYAQLDGPRCARLALPAIYAFCVLFCALPLLGLGQHQQYCPGSWCFLRMRWAQPG
GAAFSLAYAGLVALLVAAIFLCNGSVTLSLCRMYRQQKRHQGSLGPRPRTGEDEVDHLIL
LALMTVVMAVCSLPLTIRCFTQAVAPDSSSEMGDLLAFRFYAFNPILDPWVFILFRKAVF
QRLKLWVCCLCLGPAHGDSQTPLSQLASGRRDPRAPSAPVGKEGSCVPLSAWGEGQVEPL
PPTQQSSGSAVGTSSKAEASVACSLC
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| BDBM82098 |
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| n/a |
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| Name | BDBM82098 |
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| Synonyms: | 8-ISO PROSTAGLANDIN E1 | CAS_21003-46-3 | PGE1, 8-iso |
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| Type | Small organic molecule |
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| Emp. Form. | C20H34O5 |
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| Mol. Mass. | 354.481 |
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| SMILES | CCCCC[C@H](O)\C=C\C1[C@H](O)CC(=O)[C@H]1CCCCCCC(O)=O |r| |
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| Structure | 
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