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TargetThromboxane A2 receptor
LigandBDBM82213
Substrate/Competitorn/a
Ki>10000±n/a nM
CommentsPDSP_1458
Citation Armstrong, RAJones, RLWilson, NH Ligand binding to thromboxane receptors on human platelets: correlation with biological activity. Br J Pharmacol79:953-64 (1983) [PubMed]  Article
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Thromboxane A2 receptor
Name:Thromboxane A2 receptor
Synonyms:TA2R_MOUSE | Tbxa2r | Thromboxane A2
Type:Enzyme Catalytic Domain
Mol. Mass.:37114.77
Organism:MOUSE
Description:Thromboxane A2 TBXA2R MOUSE::P30987
Residue:341
Sequence:
MWPNGTSLGACFRPVNITLQERRAIASPWFAASFCALGLGSNLLALSVLAGARPGAGPRS
SFLALLCGLVLTDFLGLLVTGAIVASQHAALLDWRATDPSCRLCYFMGVAMVFFGLCPLL
LGAAMASERFVGITRPFSRPTATSRRAWATVGLVWVAAGALGLLPLLGLGRYSVQYPGSW
CFLTLGTQRGDVVFGLIFALLGSASVGLSLLLNTVSVATLCRVYHTREATQRPRDCEVEM
MVQLVGIMVVATVCWMPLLVFIMQTLLQTPPVMSFSGQLLRATEHQLLIYLRVATWNQIL
DPWVYILFRRSVLRRLHPRFSSQLQAVSLRRPPAQAMLSGP
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  Blast E-value cutoff:
BDBM82213
n/a
NameBDBM82213
Synonyms:CAS_41598-07-6 | NSC_114678 | PGD2
TypeSmall organic molecule
Emp. Form.C20H30O4
Mol. Mass.334.4498
SMILESCCCCCC(O)CC=C1C(CC=CCCCC(O)=O)C=CC1=O |w:8.7,12.11,c:20|
Structure
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