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TargetD(1A) dopamine receptor
LigandBDBM24183
Substrate/Competitorn/a
Ki>10000±n/a nM
CommentsPDSP_867
Citation Billard, WRuperto, VCrosby, GIorio, LCBarnett, A Characterization of the binding of 3H-SCH 23390, a selective D-1 receptor antagonist ligand, in rat striatum. Life Sci35:1885-93 (1984) [PubMed]  Article
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D(1A) dopamine receptor
Name:D(1A) dopamine receptor
Synonyms:DOPAMINE D1 | DRD1_RAT | Dopamine D1 high | Dopamine D1 low | Dopamine receptor | Dopamine receptor D1 | Dopamine1-like | Drd1 | Drd1a
Type:Enzyme Catalytic Domain
Mol. Mass.:49429.75
Organism:RAT
Description:P18901
Residue:446
Sequence:
MAPNTSTMDEAGLPAERDFSFRILTACFLSLLILSTLLGNTLVCAAVIRFRHLRSKVTNF
FVISLAVSDLLVAVLVMPWKAVAEIAGFWPLGPFCNIWVAFDIMCSTASILNLCVISVDR
YWAISSPFQYERKMTPKAAFILISVAWTLSVLISFIPVQLSWHKAKPTWPLDGNFTSLED
TEDDNCDTRLSRTYAISSSLISFYIPVAIMIVTYTSIYRIAQKQIRRISALERAAVHAKN
CQTTAGNGNPVECAQSESSFKMSFKRETKVLKTLSVIMGVFVCCWLPFFISNCMVPFCGS
EETQPFCIDSITFDVFVWFGWANSSLNPIIYAFNADFQKAFSTLLGCYRLCPTTNNAIET
VSINNNGAVVFSSHHEPRGSISKDCNLVYLIPHAVGSSEDLKKEEAGGIAKPLEKLSPAL
SVILDYDTDVSLEKIQPVTHSGQHST
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  Blast E-value cutoff:
BDBM24183
n/a
NameBDBM24183
Synonyms:4-amino-n-[2,3-3H]butyric acid | 4-aminobutanoic acid | Aminalon | CHEMBL96 | GABA | Gamma-Aminobutyric acid | [3H]GABA | cid_119
TypeRadiolabeled ligand
Emp. Form.C4H9NO2
Mol. Mass.103.1198
SMILESNCCCC(O)=O
Structure
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